SCHEMBL692241

SCHEMBL692241

CC(C)(C)c1ccc(CN2COC(c3cc(Cl)c(O)c(Cl)c3)=N2)cc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 3/20 0.40
HSP90AB1 P08238 3/20 0.40
AKR1C2 P52895 1/20 0.40
AKR1C1 Q04828 1/20 0.40
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
S1PR1 P21453 4/20 0.35
S1PR4 O95977 3/20 0.35
S1PR5 Q9H228 3/20 0.35
CCR9 P51686 4/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
S1PR3 Q99500 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21351756 0.66 KDM4E (0.34) ALDH1A1HTTNPSR1
SCHEMBL1114208 0.65 KDM4E (0.36) ALDH1A1CCR9OPRM1
SCHEMBL6862404 0.63 KCNH2 (0.37) ALDH1A1HTTNPSR1
SCHEMBL6321695 0.61 GABRA1 (0.52) AKR1C2AKR1C1ALDH1A1
SCHEMBL10826347 0.61 AKR1C2 (0.41) AKR1C2AKR1C1
SCHEMBL29065613 0.59 GABRA1 (0.50) AKR1C2AKR1C1ALDH1A1
SCHEMBL12891080 0.59 KCNH2 (0.48) ALDH1A1S1PR1S1PR4S1PR5
SCHEMBL28861008 0.59 HSP90AA1 (0.49) HSP90AA1HSP90AB1ALDH1A1HTTNPSR1
SCHEMBL1044315 0.59 KCNH2 (0.58) ALDH1A1
SCHEMBL6047987 0.59 KCNH2 (0.50) ALDH1A1S1PR1S1PR4S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421528-A1 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING 1,3,4-OXADIAZOLE DERIVATIVES Institute for OneWorld Health (US) 2012-02-29 EP disclosed
WO-2010123933-A1 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING 1,3,4-OXADIAZOLE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2010-10-28 WO disclosed