SCHEMBL1114208

SCHEMBL1114208

Oc1c(Cl)cc(C2=NCN(Cc3ccc(C(F)(F)F)cc3)O2)cc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
OPRL1 P41146 3/20 0.35
OPRM1 P35372 1/20 0.35
SRC P12931 1/20 0.35
PRKACA P17612 1/20 0.35
PRKACG P22612 1/20 0.35
PRKACB P22694 1/20 0.35
CHRM5 P08912 1/20 0.34
CHRM3 P20309 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
PARP1 P09874 2/20 0.34
PARP2 Q9UGN5 2/20 0.34
COMT P21964 1/20 0.33
HIF1A Q16665 1/20 0.33
EPAS1 Q99814 1/20 0.33
PHGDH O43175 1/20 0.33
CACNA1G O43497 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1114224 0.89 KDM4E (0.41) KDM4EALDH1A1
SCHEMBL1114292 0.75 MEP1B (0.36)
SCHEMBL4505012 0.68 HDAC1 (0.44) SRCPRKACAPRKACGPRKACBCCR9
SCHEMBL692241 0.65 HSP90AA1 (0.40) ALDH1A1OPRM1CCR9
SCHEMBL1114207 0.64 SRC (0.35) KDM4EALDH1A1OPRL1OPRM1SRC
SCHEMBL1114522 0.64 ALDH1A1 (0.41) KDM4EALDH1A1
SCHEMBL16856741 0.61 HDAC6 (0.47) KDM4EALDH1A1OPRL1OPRM1CHRM5
SCHEMBL4357500 0.60 HDAC3 (0.46)
SCHEMBL5600053 0.60 ALDH1A1 (0.50) KDM4EALDH1A1HIF1A
SCHEMBL15243043 0.59 HDAC6 (0.48) KDM4EALDH1A1OPRL1CHRM5CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278879-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES Institute for OneWorld Health (US) 2011-02-02 EP disclosed
WO-2009131957-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2009-10-29 WO disclosed