SCHEMBL6923115

SCHEMBL6923115

N#Cc1cccc(-c2ccc([NH])nc2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 2/20 0.53
MAP4K4 O95819 1/20 0.48
GABRG2 P18507 5/20 0.48
GABRB3 P28472 5/20 0.48
GABRA5 P31644 5/20 0.48
GABRA3 P34903 5/20 0.48
GABRA1 P14867 1/20 0.48
IDO1 P14902 2/20 0.46
CYP17A1 P05093 1/20 0.45
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
GRM5 P41594 1/20 0.45
XDH P47989 1/20 0.44
SLC22A12 Q96S37 1/20 0.44
PLG P00747 1/20 0.44
PLAU P00749 1/20 0.44
USP30 Q70CQ3 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4021783 0.80 CYP11B2 (0.56) CLK4MAP4K4GABRG2GABRB3GABRA5
SCHEMBL5562910 0.80 MAP4K4 (0.62) CLK4MAP4K4GABRG2GABRB3GABRA5
SCHEMBL3266198 0.80 CLK4 (0.53) CLK4MAP4K4GABRG2GABRB3GABRA5
SCHEMBL3881340 0.80 CLK4 (0.53) CLK4MAP4K4GABRG2GABRB3GABRA5
SCHEMBL2154026 0.78 CLK4 (0.65) CLK4MAP4K4GABRG2GABRB3GABRA5
SCHEMBL18223984 0.76 SYK (0.53) CLK4MAP4K4GABRG2GABRB3GABRA5
SCHEMBL5562878 0.76 GABRG2 (0.52) CLK4MAP4K4GABRG2GABRB3GABRA5
SCHEMBL5558730 0.76 HSD17B1 (0.60) CLK4MAP4K4GABRG2GABRB3GABRA5
SCHEMBL5557633 0.76 CLK4 (0.54) CLK4MAP4K4GABRG2GABRB3GABRA5
SCHEMBL14224867 0.76 CLK4 (0.49) CLK4MAP4K4GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441719-A1 N-SUBSTITUTED PYRROLIDIN DERIVATIVES AS DIPEPTIDYL PEPTIDASE IV INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2004-08-04 EP disclosed
WO-2003037327-A1 N-SUBSTITUTED PYRROLIDIN DERIVATIVES AS DIPEPTIDYL PEPTIDASE IV INHIBITORS F. HOFFMANN-LA-ROCHE AG (CH) 2003-05-08 WO disclosed