SCHEMBL6923362

SCHEMBL6923362

COP(=O)(O)[C@H](C)NC(=O)OCc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KYNU Q16719 1/20 0.57
ELANE P08246 2/20 0.56
ATM Q13315 1/20 0.53
PRTN3 P24158 2/20 0.53
ACE2 Q9BYF1 1/20 0.52
LAP3 P28838 1/20 0.51
CTSK P43235 3/20 0.51
TACR1 P25103 1/20 0.51
CTRB1 P17538 2/20 0.50
MME P08473 1/20 0.50
ECE1 P42892 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6923368 1.00 KYNU (0.57) KYNUELANEATMPRTN3ACE2
SCHEMBL12942520 0.87 ELANE (0.61) KYNUELANEATMPRTN3ACE2
SCHEMBL11567174 0.87 ELANE (0.60) KYNUELANEATMPRTN3ACE2
SCHEMBL4163321 0.87 ELANE (0.60) KYNUELANEATMPRTN3ACE2
SCHEMBL8740045 0.87 ELANE (0.60) KYNUELANEATMPRTN3ACE2
SCHEMBL5076528 0.86 ELANE (0.67) KYNUELANEATMPRTN3ACE2
SCHEMBL8587097 0.86 ELANE (0.59) KYNUELANEATMPRTN3ACE2
SCHEMBL7397375 0.84 ECE1 (0.59) KYNUACE2LAP3TACR1CTRB1
SCHEMBL14981588 0.84 ALDH1A1 (0.56) KYNUELANEATMPRTN3ACE2
SCHEMBL10955973 0.82 KYNU (0.56) KYNUELANEPRTN3ACE2MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6737416-B2 THROMBOLYTIC AGENT HAVING HIGHER SAFETY MEIJI SEIKA KAISHA LTD. (JP) 2004-05-18 US disclosed
US-20030119787-A1 Phosphonic acid derivative having inhibitory activity against carboxypeptidase B MEIJI SEIKA KAISHA LTD. (JP) 2003-06-26 US disclosed
US-6576627-B1 Such as 7-amino-2-((2-methyl-1-(3-phenylpropanoylamino)-propyl)hydroxyphosphinoyl) -methylheptanoic acid; thrombotic disease MEIJI SEIKA KAISHA LTD. (JP) 2003-06-10 US disclosed
EP-1152004-B1 Phosphonic acid derivatives having carboxypeptidase B inhibitory action MEIJI SEIKA KAISHA (JP) 2003-05-07 EP disclosed
EP-1174434-A1 Phosphonic acid derivative having inhibitory activity against carboxypeptidase B MEIJI SEIKA KAISHA LTD. (JP) 2002-01-23 EP disclosed
EP-1152004-A1 PHOSPHONIC ACID DERIVATIVES HAVING CARBOXYPEPTIDASE B INHIBITORY ACTIVITY MEIJI SEIKA KAISHA LTD. (JP) 2001-11-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030119787-A1 Phosphonic acid derivative having inhibitory activity against carboxypeptidase B CPB1, RNPEP, CPN1 KYNU 3943/4885ELANE 173/4885ATM 4673/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.