SCHEMBL6924481

SCHEMBL6924481

CCCS(=O)(=O)N1CCN(c2ccc(-c3nc(-c4ccc(Cl)cc4)c[nH]3)cn2)CC1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.49
HSD17B10 Q99714 1/20 0.49
GPR119 Q8TDV5 9/20 0.41
CNR2 P34972 2/20 0.41
CNR1 P21554 1/20 0.41
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
SUV39H2 Q9H5I1 1/20 0.39
SMO Q99835 1/20 0.39
KMT2A Q03164 1/20 0.38
GLA P06280 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
DGAT1 O75907 1/20 0.38
KCNH2 Q12809 1/20 0.38
ADK P55263 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6926962 0.88 RET (0.47) GPR119CNR2SMOKMT2AL3MBTL1
SCHEMBL6923696 0.83 RET (0.43) KDM4ECNR2DGAT1KCNH2
SCHEMBL6927440 0.82 HRH4 (0.51) CNR2KMT2ADGAT1KCNH2
SCHEMBL6920570 0.78 RET (0.42) CNR2ALDH1A1DGAT1KCNH2
SCHEMBL6929138 0.78 FAAH (0.46) KDM4EHSD17B10GPR119CNR2ALDH1A1
SCHEMBL6924758 0.76 PKM (0.41) KDM4EALDH1A1SMOL3MBTL1DGAT1
SCHEMBL6924750 0.76 CNR2 (0.46) CNR2
SCHEMBL6923619 0.75 DRD3 (0.47)
SCHEMBL6926613 0.75 TDO2 (0.41) KDM4EGPR119ALDH1A1L3MBTL1DGAT1
SCHEMBL6923542 0.75 MEN1 (0.44) KDM4EGPR119ALDH1A1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514966-B2 Neuropeptide Y antagonists such as 2-chloro-5-(4-(3,4-dich loro-phenyl)-1H-imidazol-2-yl)-pyridine PFIZER INC. 2003-02-04 US disclosed
US-6355635-B1 IMIDAZOLEBENZENE, IMIDAZOLEPYRIDINE COMPOUNDS FOR TREATMENT OF OBESITY PFIZER INC. 2002-03-12 US disclosed
US-20010039277-A1 Compounds for the treatment of obesity ELLIOTT RICHARD L (US) 2001-11-08 US disclosed
WO-2000066578-A1 COMPOUNDS FOR THE TREATMENT OF OBESITY PFIZER PRODUCTS INC. (US) 2000-11-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010039277-A1 Compounds for the treatment of obesity NPY1R, NPY4R, NPY2R KDM4E 1926/4885HSD17B10 800/4885GPR119 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.