SCHEMBL6926962

SCHEMBL6926962

CS(=O)(=O)N1CCN(c2ccc(-c3nc(-c4ccc(Cl)cc4)c[nH]3)cn2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 2/20 0.47
CNR2 P34972 1/20 0.44
IKBKB O14920 1/20 0.43
KDR P35968 1/20 0.42
ETV6 P41212 1/20 0.42
LRRK2 Q5S007 1/20 0.41
GPR119 Q8TDV5 1/20 0.40
KMT2A Q03164 1/20 0.40
ALOX5AP P20292 1/20 0.40
KCNH2 Q12809 2/20 0.40
SMO Q99835 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
DGAT1 O75907 1/20 0.40
ADK P55263 1/20 0.40
ABL1 P00519 1/20 0.40
BCR P11274 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
MAPK1 P28482 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6924481 0.88 KDM4E (0.49) CNR2GPR119KMT2AKCNH2SMO
SCHEMBL6927440 0.85 HRH4 (0.51) RETCNR2KMT2AKCNH2DGAT1
SCHEMBL6923696 0.82 RET (0.43) RETCNR2KDRKCNH2DGAT1
SCHEMBL6929138 0.82 FAAH (0.46) RETCNR2GPR119KMT2AKCNH2
SCHEMBL6920570 0.80 RET (0.42) RETCNR2KCNH2DGAT1MGLL
SCHEMBL2155271 0.78 GPR119 (0.59) RETCNR2GPR119KMT2ASMO
SCHEMBL6926613 0.78 TDO2 (0.41) RETGPR119L3MBTL1DGAT1MAPK1
SCHEMBL6923542 0.78 MEN1 (0.44) GPR119KMT2AL3MBTL1ADKMAPK1
SCHEMBL6927606 0.76 KDM4E (0.55) KMT2AL3MBTL1ABL1BCRMAPK1
SCHEMBL6924758 0.75 PKM (0.41) RETSMOL3MBTL1DGAT1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514966-B2 Neuropeptide Y antagonists such as 2-chloro-5-(4-(3,4-dich loro-phenyl)-1H-imidazol-2-yl)-pyridine PFIZER INC. 2003-02-04 US disclosed
US-6355635-B1 IMIDAZOLEBENZENE, IMIDAZOLEPYRIDINE COMPOUNDS FOR TREATMENT OF OBESITY PFIZER INC. 2002-03-12 US disclosed
US-20010039277-A1 Compounds for the treatment of obesity ELLIOTT RICHARD L (US) 2001-11-08 US disclosed
WO-2000066578-A1 COMPOUNDS FOR THE TREATMENT OF OBESITY PFIZER PRODUCTS INC. (US) 2000-11-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010039277-A1 Compounds for the treatment of obesity NPY1R, NPY4R, NPY2R RET 1562/4885CNR2 122/4885IKBKB 770/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.