SCHEMBL6925924

SCHEMBL6925924

CSc1ccc(-c2nc3c(Cl)nc4ccccc4c3n2CCC2CCN(C(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 3/20 0.44
KDM4E B2RXH2 1/20 0.40
PKM P14618 1/20 0.40
HPGDS O60760 1/20 0.37
GAA P10253 1/20 0.37
THRB P10828 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
LMNA P02545 2/20 0.37
MAPT P10636 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
CCR5 P51681 1/20 0.37
TP53 P04637 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
GBA1 P04062 1/20 0.36
PTGER4 P35408 1/20 0.36
BRD4 O60885 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6838678 0.93 KDM4E (0.43) GPR119KDM4EPKMHPGDSTHRB
SCHEMBL6927289 0.82 GBA1 (0.40) GPR119KDM4EPKMTHRBLMNA
SCHEMBL6833883 0.82 KDM4E (0.42) GPR119KDM4EPKMHPGDSTHRB
SCHEMBL6927222 0.81 ACKR3 (0.45) THRBSMN1; SMN2MAPTTP53MEN1
SCHEMBL6838661 0.81 CETP (0.42) GPR119KDM4EPKMHPGDSLMNA
SCHEMBL6837673 0.79 HPGDS (0.47) GPR119KDM4EPKMHPGDSTHRB
SCHEMBL6928754 0.79 CKS1B (0.38) GPR119PTGER4BRD4
SCHEMBL6929719 0.79 PTGER4 (0.37) PTGER4BRD4
SCHEMBL6927078 0.78 KDM4E (0.45) GPR119KDM4EPKM
SCHEMBL6926356 0.76 ALDH1A1 (0.37) KDM4EGAASMN1; SMN2LMNATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6518265-B1 1H-imidazopyridine derivatives HOKURIKU SEIYAKU CO., LTD. (JP) 2003-02-11 US disclosed
EP-1104764-A1 1H-IMIDAZOPYRIDINE DERIVATIVES HOKURIKU SEIYAKU CO., LTD. (JP) 2001-06-06 EP disclosed