SCHEMBL6926692

SCHEMBL6926692

O=CN1Cc2cccc(F)c2C1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRAP1 Q12931 4/20 0.42
HSP90B1 P14625 2/20 0.42
DPP8 Q6V1X1 2/20 0.40
DPP9 Q86TI2 2/20 0.40
DPP7 Q9UHL4 2/20 0.40
TIPARP Q7Z3E1 1/20 0.40
TSHR P16473 1/20 0.39
KCNH2 Q12809 3/20 0.38
TMEM97 Q5BJF2 3/20 0.38
SIGMAR1 Q99720 3/20 0.38
IP6K1 Q92551 1/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
PKM P14618 1/20 0.35
PKLR P30613 1/20 0.35
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22730588 0.84 PDE4D (0.41) TRAP1HSP90B1DPP8DPP9DPP7
SCHEMBL12765385 0.78 CYP1A2 (0.42) TRAP1TSHRKMT2AMEN1
SCHEMBL23505868 0.78 TRAP1 (0.42) TRAP1
SCHEMBL1301328 0.77 NOTUM (0.44) TRAP1HSP90B1KMT2AMEN1PKM
SCHEMBL29008582 0.75 ALDH1A1 (0.34) KMT2AMEN1PKMDRD2
SCHEMBL23505873 0.74 TRPA1 (0.42) TSHRKCNH2SIGMAR1KMT2AMEN1
SCHEMBL25234740 0.74 RAB9A (0.34) L3MBTL1
SCHEMBL14626026 0.74 PDE4D (0.47) TRAP1HSP90B1TIPARPDRD2DRD3
SCHEMBL30970493 0.74 RAB9A (0.34) L3MBTL1
SCHEMBL8217297 0.74 TRAP1 (0.53) TRAP1HSP90B1DPP8DPP9DPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011109551-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA INC. (US) 2011-09-09 WO disclosed
EP-2305698-A2 Macrocyclic inhibitors of Hepatitis C virus replication Intermune, Inc. (US) 2011-04-06 EP disclosed
WO-2007015824-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2007-02-08 WO disclosed