SCHEMBL6928014

SCHEMBL6928014

COC(Oc1cccc([N+](=O)[O-])c1)C(=O)Cl

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
TSHR P16473 2/20 0.49
F2 P00734 1/20 0.46
LMNA P02545 3/20 0.45
MAOB P27338 2/20 0.45
CHRNB2 P17787 1/20 0.45
CHRNA4 P43681 1/20 0.45
MAPT P10636 3/20 0.44
MEN1 O00255 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
MAOA P21397 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6921768 0.87 ALDH1A1 (0.49) ALDH1A1TSHRF2LMNAMAOB
SCHEMBL9770479 0.84 MEN1 (0.49) ALDH1A1LMNAMAOBMAPTMEN1
SCHEMBL10638083 0.79 ALDH1A1 (0.48) ALDH1A1TSHRF2LMNAMAOB
SCHEMBL16097479 0.78 LMNA (0.48) ALDH1A1TSHRF2LMNAMAOB
SCHEMBL20299326 0.77 TSHR (0.52) ALDH1A1TSHRF2LMNAMAOB
SCHEMBL7671999 0.77 TSHR (0.55) ALDH1A1TSHRF2LMNACHRNB2
SCHEMBL16764355 0.76 F2 (0.57) ALDH1A1TSHRF2LMNAMAPT
SCHEMBL6920987 0.76 ALDH1A1 (0.42) ALDH1A1CHRNB2CHRNA4MAPTMEN1
SCHEMBL657614 0.75 ALDH1A1 (0.59) ALDH1A1F2LMNAMAPTMEN1
SCHEMBL27679166 0.75 ALDH1A1 (0.59) ALDH1A1F2LMNAMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001766-B1 COMPOUNDS FOR THE TREATMENT OF CCR5-MEDIATED DISEASES SMITHKLINE BEECHAM CORP (US) 2003-04-09 EP disclosed
US-6515027-B1 Ligands, agonists or antagonists, of the CC chemokine receptor CC-CKR5 SMITHKLINE BEECHAM CORP. 2003-02-04 US disclosed
EP-1001766-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2001-04-04 EP disclosed
EP-1001766-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999001127-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-01-14 WO disclosed