SCHEMBL8562859

SCHEMBL8562859

CCc1c(Sc2ccccc2)nc(C)n1COCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
VCP P55072 2/20 0.35
TSHR P16473 2/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
LMNA P02545 2/20 0.34
TNF P01375 1/20 0.33
L3MBTL1 Q9Y468 3/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
POLB P06746 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NPSR1 Q6W5P4 2/20 0.32
PRNP P04156 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
PPARG P37231 1/20 0.32
HTT P42858 1/20 0.32
NCOA2 Q15596 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567515 0.74 VCP (0.41) ALDH1A1VCPTSHRSMN1; SMN2L3MBTL1
SCHEMBL8560120 0.74 ALDH1A1 (0.38) ALDH1A1VCPTSHRSMN1; SMN2LMNA
SCHEMBL8562572 0.72 ALDH1A1 (0.38) ALDH1A1VCPTSHRSMN1; SMN2L3MBTL1
SCHEMBL9050612 0.72 ALDH1A1 (0.40) ALDH1A1VCPTSHRSMN1; SMN2LMNA
SCHEMBL8562834 0.71 ALDH1A1 (0.44) ALDH1A1VCPTSHRSMN1; SMN2LMNA
SCHEMBL8568227 0.71 ALDH1A1 (0.39) ALDH1A1VCPTSHRSMN1; SMN2LMNA
SCHEMBL7854175 0.69 ALDH1A1 (0.40) ALDH1A1VCPTSHRSMN1; SMN2TNF
SCHEMBL8567153 0.68 CSNK1D (0.42) ALDH1A1TSHRSMN1; SMN2LMNAL3MBTL1
SCHEMBL9051616 0.68 ALDH1A1 (0.40) ALDH1A1VCPTSHRLMNAL3MBTL1
SCHEMBL8562868 0.68 ALDH1A1 (0.36) ALDH1A1SMN1; SMN2LMNATNFL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0552060-B1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO (JP) 1998-11-18 EP disclosed
EP-0700911-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1996-03-13 EP disclosed
US-5472965-A Useful for treatment of retrovirus infections; less toxic SHIONOGI & CO., LTD. (JP) 1995-12-05 US disclosed
US-5326780-A Acquired immunodeficiency syndrome SHIONOGI & CO., LTD. (JP) 1994-07-05 US disclosed
EP-0552060-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1993-07-21 EP disclosed