SCHEMBL6928397

SCHEMBL6928397

CC(C)(C)[Si](C)(C)OCc1ccc(C#N)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.42
CYP11B1 P15538 12/20 0.38
CYP11B2 P19099 12/20 0.38
DAO P14920 2/20 0.38
CACNA1H O95180 3/20 0.37
CNR1 P21554 1/20 0.36
RORC P51449 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18314460 0.84 TRPV4 (0.38) TRPV4
SCHEMBL8143451 0.83 SNCA (0.37)
SCHEMBL7715279 0.81 DAO (0.43) TRPV4CYP11B1CYP11B2DAOCACNA1H
SCHEMBL19387960 0.79 TRPV4 (0.47) TRPV4CYP11B1CYP11B2DAOCACNA1H
SCHEMBL4074377 0.78 APLNR (0.33)
SCHEMBL2596478 0.78 ALDH1A1 (0.36)
SCHEMBL8003064 0.77 TRPV4 (0.40) TRPV4CYP11B1CYP11B2DAOCNR1
SCHEMBL31605567 0.77 TRPV4 (0.52) TRPV4CYP11B1CYP11B2DAOCNR1
SCHEMBL16892292 0.77 TRPV4 (0.52) TRPV4CYP11B1CYP11B2DAOCNR1
SCHEMBL481069 0.76 CACNA1H (0.34) CYP11B1CYP11B2CACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1135023-A4 AMINOBENZISOXAZOLE COMPOUNDS AND LIBRARIES THEREOF LILLY CO ELI (US) 2003-03-05 EP disclosed
EP-1135023-A1 AMINOBENZISOXAZOLE COMPOUNDS AND LIBRARIES THEREOF ELI LILLY AND COMPANY (US) 2001-09-26 EP disclosed
WO-2000027199-A1 AMINOBENZISOXAZOLE COMPOUNDS AND LIBRARIES THEREOF ELI LILLY AND COMPANY (US) 2000-05-18 WO disclosed