SCHEMBL6930355

SCHEMBL6930355

NOC(Cl)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 14/20 0.50
TDO2 P48775 11/20 0.50
TSHR P16473 1/20 0.50
IDO2 Q6ZQW0 3/20 0.47
DPP4 P27487 2/20 0.43
F2 P00734 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3774968 0.78 TSHR (0.55) IDO1TDO2TSHRIDO2DPP4
SCHEMBL7915804 0.78 TSHR (0.55) IDO1TDO2TSHRIDO2DPP4
SCHEMBL13278769 0.74 TSHR (0.50) IDO1TDO2TSHRIDO2DPP4
SCHEMBL11666583 0.74 TSHR (0.50) IDO1TDO2TSHRIDO2DPP4
SCHEMBL105848 0.74 TSHR (0.50) TSHRDPP4F2
SCHEMBL7099520 0.74 TSHR (0.50) IDO1TDO2TSHRIDO2DPP4
SCHEMBL27256310 0.74 TSHR (0.50) TSHRDPP4F2
SCHEMBL15974014 0.74 TSHR (0.50) TSHRDPP4F2
SCHEMBL98309 0.72 IDO1 (0.74) IDO1TDO2IDO2
SCHEMBL6157714 0.72 TSHR (0.48) TSHRDPP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697193-A1 SUBSTITUTED 5-(CYCLOHEX-2-EN-1-YL)-PENTA-2,4-DIENES AND 5-(CYCLOHEX-2-EN-1-YL)-PENT-2-EN-4-INES AS ACTIVE AGENTS AGAINST ABIOTIC STRESS IN PLANTS Bayer Intellectual Property GmbH (DE) 2014-02-19 EP disclosed
WO-2012139890-A1 SUBSTITUTED 5-(CYCLOHEX-2-EN-1-YL)-PENTA-2,4-DIENES AND 5-(CYCLOHEX-2-EN-1-YL)-PENT-2-EN-4-INES AS ACTIVE AGENTS AGAINST ABIOTIC STRESS IN PLANTS BAYER CROPSCIENCE AG (DE) 2012-10-18 WO disclosed
EP-0835279-B1 IMPROVED SURFACE TREATMENT OF POLYMERS COMMW SCIENT ANDINDUSTRIAL RES (AU) 2003-12-17 EP disclosed
EP-1196451-A4 SURFACE MODIFICATION OF VULCANISED RUBBER OBJECTS COMMW SCIENT IND RES ORG (AU) 2002-10-24 EP disclosed
US-20020074696-A1 Surface modification of vulcanised rubber objects COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2002-06-20 US disclosed
CN-1085990-C Improved surface treatment of polymers COMMW SCIENT IND RES ORG (AU) 2002-06-05 CN disclosed
EP-1196451-A1 SURFACE MODIFICATION OF VULCANISED RUBBER OBJECTS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2002-04-17 EP disclosed
WO-2000053638-A1 SURFACE MODIFICATION OF VULCANISED RUBBER OBJECTS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2000-09-14 WO disclosed
US-5922161-A OXIDIZING PART OF THE SURFACE OF THE POLYMER; TREATING WITH A MULTIFUNCTIONAL AMINE-CONTAINING ORGANIC COMPOUND; BINDING ADHESIVES, COATINGS, PAINTS; MEDICAL EQUIPMENT; BONDING STRENGTH; STORAGE STABILITY COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 1999-07-13 US disclosed
EP-0835279-A4 IMPROVED SURFACE TREATMENT OF POLYMERS COMMW SCIENT IND RES ORG (AU) 1999-02-17 EP disclosed
CN-1192224-A Improved polymer surface treatment process COMMW SCIENT IND RES ORG (AU) 1998-09-02 CN disclosed
EP-0835279-A1 IMPROVED SURFACE TREATMENT OF POLYMERS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 1998-04-15 EP disclosed
WO-1997002310-A1 IMPROVED SURFACE TREATMENT OF POLYMERS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 1997-01-23 WO disclosed