SCHEMBL6930673

SCHEMBL6930673

CC1C=Cc2c(-c3ccccc3)cccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
PDCD1 Q15116 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
BRD4 O60885 1/20 0.34
ALDH1A1 P00352 3/20 0.33
HSD17B10 Q99714 2/20 0.33
HPGD P15428 1/20 0.33
BCL2L1 Q07817 1/20 0.33
CYP2A6 P11509 1/20 0.33
MAPK1 P28482 1/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
HTR7 P34969 3/20 0.32
HTR1A P08908 2/20 0.32
HTR2B P41595 2/20 0.32
TMEM97 Q5BJF2 2/20 0.32
SIGMAR1 Q99720 2/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31108156 1.00 CHRNB2 (0.36) CHRNB2CHRNA4PDCD1CD274BRD4
SCHEMBL2973463 0.81 ALDH1A1 (0.34) ALDH1A1MAPK1
SCHEMBL27448311 0.78 CHRNB2 (0.36) CHRNB2CHRNA4PDCD1CD274BRD4
Hydrochloric Acid SCHEMBL5184845 0.78 CHRNB2 (0.36) CHRNB2CHRNA4PDCD1CD274BRD4
SCHEMBL28325453 0.78 CHRNB2 (0.36) CHRNB2CHRNA4PDCD1CD274BRD4
Fluoride SCHEMBL5183962 0.78 CHRNB2 (0.36) CHRNB2CHRNA4PDCD1CD274BRD4
SCHEMBL5860378 0.78 CHRNB2 (0.36) CHRNB2CHRNA4PDCD1CD274BRD4
SCHEMBL4059907 0.78 MGLL (0.38) CHRNB2CHRNA4PDCD1CD274BRD4
SCHEMBL28814578 0.77 CHRNB2 (0.33) CHRNB2CHRNA4PDCD1CD274BRD4
SCHEMBL7870640 0.77 ADRA2A (0.33) CHRNB2CHRNA4PDCD1CD274BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1027314-A4 COUPLING REACTIONS OF 2-SUBSTITUTED, 7-HALOINDENES WITH ARYL SUBSTITUENTS TO PRODUCE METALLOCENE CATALYST LIGANDS BOULDER SCIENT CO (US) 2003-03-19 EP claimed
US-6465700-B1 E.G., 2-METHYL-7-CHLOROINDENE. BOULDER SCIENTIFIC COMPANY 2002-10-15 US claimed
EP-1027314-A1 COUPLING REACTIONS OF 2-SUBSTITUTED, 7-HALOINDENES WITH ARYL SUBSTITUENTS TO PRODUCE METALLOCENE CATALYST LIGANDS BOULDER SCIENTIFIC COMPANY (US) 2000-08-16 EP claimed
WO-2000007968-A1 COUPLING REACTIONS OF 2-SUBSTITUTED, 7-HALOINDENES WITH ARYL SUBSTITUENTS TO PRODUCE METALLOCENE CATALYST LIGANDS BOULDER SCIENTIFIC COMPANY (US) 2000-02-17 WO claimed
CN-117004966-A Synthesis method of benzoferrocene phosphine oxide compound 中国科学院大连化学物理研究所 2023-11-07 CN disclosed