SCHEMBL6930675

SCHEMBL6930675

Cc1ccc(NC(C)C2CC2)cc1O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
MEN1 O00255 1/20 0.42
CYP3A4 P08684 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
TRPA1 O75762 1/20 0.42
PTGS1 P23219 1/20 0.42
CACNA1C Q13936 1/20 0.42
IDH1 O75874 3/20 0.40
ALDH1A1 P00352 2/20 0.40
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
LMNA P02545 2/20 0.37
EPHX2 P34913 1/20 0.36
TSHR P16473 1/20 0.36
CASP1 P29466 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL453729 0.78 TRPA1 (0.50) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL95127 0.77 TRPA1 (0.48) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL6933453 0.77 TRPA1 (0.48) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL6932118 0.72 ALDH1A1 (0.59) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL6928569 0.70 CYP1A2 (0.57) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL7688086 0.70 CYP1A2 (0.57) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL6930690 0.70 ALDH1A1 (0.50) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL455968 0.69 GFER (0.44) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL6928541 0.69 GFER (0.47) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL6932279 0.69 CYP2D6 (0.44) CYP1A2CYP2D6CYP2C9CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1224374-C Novel couplers for oxidative hair dyeing P & G CLAIROL INC (US) 2005-10-26 CN disclosed
CN-1477948-A Novel couplers for oxidative hair dyeing P&G克莱罗尔公司 2004-02-25 CN disclosed
EP-1363587-A1 NOVEL COUPLER FOR USE IN OXIDATIVE HAIR DYEING P&G-Clairol, Inc. (US) 2003-11-26 EP disclosed
US-6409773-B1 AMINOPHENOL COUPLERS CLAIROL INCORPORATED 2002-06-25 US disclosed
WO-2002047635-A1 NOVEL COUPLER FOR USE IN OXIDATIVE HAIR DYEING P&G-CLAIROL, INC. (US) 2002-06-20 WO disclosed