SCHEMBL6933717

SCHEMBL6933717

CCNC(=O)Nc1ncc(C)c(C(F)(F)F)n1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
JUN P05412 2/20 0.41
NFKB1 P19838 2/20 0.41
NFKB2 Q00653 2/20 0.41
RELA Q04206 2/20 0.41
KDM4E B2RXH2 1/20 0.40
SORT1 Q99523 1/20 0.39
ABL1 P00519 2/20 0.39
MKNK2 Q9HBH9 1/20 0.39
MAPK1 P28482 4/20 0.38
PIK3CA P42336 4/20 0.38
PIK3CD O00329 1/20 0.37
MAPK8 P45983 2/20 0.37
MAPK9 P45984 2/20 0.37
MAPK10 P53779 2/20 0.37
MAPK14 Q16539 1/20 0.37
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29639807 0.82 NFKB1 (0.42) JUNNFKB1NFKB2RELAKDM4E
SCHEMBL6933248 0.75 MAPK1 (0.46) MAPK1PIK3CAMAPK8MAPK9MAPK10
SCHEMBL6933431 0.73 ABL1 (0.48) ABL1MAPK1
SCHEMBL9885815 0.68 MAPT (0.56) KDM4E
SCHEMBL19416867 0.67 RAB9A (0.62) MAPK1PIK3CAMAPK8MAPK9MAPK10
SCHEMBL10955770 0.66 MKNK1 (0.45) ABL1MKNK2
SCHEMBL24703391 0.66 PIK3CA (0.54) ABL1MAPK1PIK3CA
SCHEMBL11017429 0.66 KDM4E (0.37) NFKB1KDM4ESORT1
SCHEMBL6936291 0.66 KDM4E (0.55) KDM4EPIK3CAPIK3CD
SCHEMBL29693635 0.66 KDM4E (0.37) NFKB1KDM4ESORT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011114275-A1 SPIROCYCLIC COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS AND DIAGNOSTIC PROBES UNIVERSITY OF BASEL (CH) 2011-09-22 WO disclosed