SCHEMBL6938642

SCHEMBL6938642

COc1cccc(CN2CSC(CCO)=C2C)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
SIGMAR1 Q99720 2/20 0.45
CMA1 P23946 1/20 0.44
LPO P22079 1/20 0.42
PKM P14618 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3848581 0.99 ALDH1A1 (0.45) ALDH1A1KDM4ESIGMAR1CMA1LPO
SCHEMBL4252730 0.82 ALDH1A1 (0.43) ALDH1A1KDM4ESIGMAR1MAPTTHRB
Hydrochloric Acid SCHEMBL313570 0.80 ALDH1A1 (0.43) ALDH1A1KDM4ESIGMAR1MAPTTHRB
Bromide SCHEMBL3846883 0.78 CA12 (0.45) ALDH1A1KDM4EMAPTTP53
SCHEMBL31081822 0.72 SIGMAR1 (0.52) ALDH1A1KDM4ESIGMAR1CMA1LPO
SCHEMBL43521 0.72 TAAR1 (0.67) SIGMAR1HRH3TAAR1
Alcohol SCHEMBL5332610 0.69 TAAR1 (0.62) SIGMAR1HRH3TAAR1
Hydrochloric Acid SCHEMBL648278 0.68 SIRT2 (0.36) SIGMAR1SIRT2SIRT1
SCHEMBL27298114 0.67 SIGMAR1 (0.73) ALDH1A1KDM4ESIGMAR1PKMHRH3
SCHEMBL81474 0.66 CHRM2 (0.63) SIGMAR1HDAC1HDAC6HRH3TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808163-B1 USE OF THIAZOLIUM COMPOUNDS FOR PREVENTING AND REVERSING THE FORMATION OF ADVANCED GLYCOSYLATION ENDPRODUCTS ALTEON INC (US) 2003-07-23 EP claimed
US-6440749-B1 ADMINISTERING A THIAZOLE COMPOUND ALTEON. INC. 2002-08-27 US claimed