SCHEMBL6938929

SCHEMBL6938929

CN(C)C(c1ccc(Br)cc1)C1CCCCC1=O

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.50
LMNA P02545 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
ALDH1A1 P00352 3/20 0.44
CA1 P00915 4/20 0.40
POLB P06746 3/20 0.38
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6934444 0.85 ALDH1A1 (0.44) MAPTLMNANPSR1ALDH1A1CA1
SCHEMBL6942334 0.85 MAPT (0.50) MAPTLMNANPSR1ALDH1A1CA1
SCHEMBL5375903 0.85 CA1 (0.55) MAPTLMNANPSR1ALDH1A1CA1
SCHEMBL11794387 0.84 CA1 (0.54) MAPTLMNANPSR1ALDH1A1CA1
SCHEMBL6939750 0.82 TSHR (0.42) MAPTLMNANPSR1ALDH1A1CA1
SCHEMBL6940543 0.82 ALDH1A1 (0.41) ALDH1A1CA1
SCHEMBL6940261 0.79 SLC6A3 (0.44) MAPTLMNAALDH1A1CA1KDM4E
SCHEMBL6937407 0.78 MAPT (0.60) MAPTLMNANPSR1ALDH1A1CA1
SCHEMBL6677707 0.77 MAPT (0.42) MAPTLMNANPSR1ALDH1A1CA1
SCHEMBL6162885 0.77 ALDH1A1 (0.40) MAPTLMNANPSR1ALDH1A1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1043307-B1 3-amino-3-arylpropan-1-ol-derivates, their preparation and their use GRUENENTHAL GMBH (DE) 2003-06-04 EP disclosed
US-6410790-B1 ANALGESICS GRUENENTHAL GMBH (DE) 2002-06-25 US disclosed
EP-1043307-A2 3-amino-3-arylpropan-1-ol-derivates, their preparation and their use Grünenthal GmbH (DE) 2000-10-11 EP disclosed