SCHEMBL6940902

SCHEMBL6940902

CN(C(=O)NN[C@@H](CC(=O)O)C(N)=O)C(=O)c1cccc(CNC(=N)N)c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEP1B Q16820 2/20 0.40
PPARG P37231 2/20 0.38
ITGB3 P05106 5/20 0.36
ITGAV P06756 4/20 0.36
ITGB1 P05556 1/20 0.36
ITGA5 P08648 1/20 0.36
MDM2 Q00987 1/20 0.36
LIPG Q9Y5X9 1/20 0.35
F10 P00742 1/20 0.34
ROCK2 O75116 1/20 0.34
PRSS1 P07477 1/20 0.34
TMPRSS15 P98073 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
FNTA P49354 2/20 0.34
FNTB P49356 2/20 0.34
NR1H4 Q96RI1 1/20 0.34
HPGDS O60760 1/20 0.34
ITGA2B P08514 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6938684 0.84 ITGB3 (0.43) ITGB3ITGAVMEN1KMT2AITGA2B
SCHEMBL7878241 0.81 KCNA5 (0.37) ITGB3PRSS1TMPRSS15ITGA2B
SCHEMBL6937428 0.77 ITGB3 (0.40) ITGB3PRSS1TMPRSS15ITGA2B
SCHEMBL6939377 0.74 SELP (0.36) PPARGITGB3FNTAFNTBNR1H4
SCHEMBL7879657 0.74 ABCC1 (0.39) ITGB3PRSS1TMPRSS15KMT2AITGA2B
SCHEMBL6938012 0.70 NPY4R (0.32)
SCHEMBL20487535 0.70 NR1H4 (0.56) MEP1BF10KMT2AFNTAFNTB
SCHEMBL7878251 0.70 PRSS1 (0.35) ITGB3ITGAVPRSS1TMPRSS15ITGA2B
Hydrochloric Acid SCHEMBL7327435 0.69 NR1H4 (0.55) MEP1BF10KMT2AFNTAFNTB
SCHEMBL30940553 0.69 F10 (0.60) MEP1BF10ROCK2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326403-B1 CARDIOVASCULAR DISORDERS MERCK PATENT GESELLSCHAFT MIT (DE) 2001-12-04 US claimed
EP-1097127-B1 DIACYLHYDRAZINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2003-03-12 EP disclosed
US-6326403-B1 CARDIOVASCULAR DISORDERS MERCK PATENT GESELLSCHAFT MIT (DE) 2001-12-04 US disclosed