SCHEMBL6938012

SCHEMBL6938012

CN(C(=O)CCCCNC(=N)N)C(=O)NN[C@@H](CC(=O)O)C(N)=O

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NPY4R P50391 4/20 0.32
NPY5R Q15761 4/20 0.32
NPY1R P25929 3/20 0.32
NPY2R P49146 1/20 0.32
EPHX2 P34913 2/20 0.31
SIRT5 Q9NXA8 1/20 0.30
ADRA1A P35348 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6937672 0.77 EPHX2 (0.37) NPY4RNPY5RNPY1RNPY2REPHX2
SCHEMBL6940902 0.70 MEP1B (0.40)
SCHEMBL7878241 0.70 KCNA5 (0.37)
SCHEMBL7416968 0.68 NPY4R (0.36) NPY4RNPY5RNPY1RNPY2R
SCHEMBL6937428 0.68 ITGB3 (0.40)
SCHEMBL7878251 0.68 PRSS1 (0.35)
SCHEMBL7879657 0.68 ABCC1 (0.39)
SCHEMBL2107302 0.67 PRMT1 (0.59) ADRA1A
SCHEMBL23732364 0.66 KDM4A (0.41) EPHX2ADRA1A
Trifluoroacetic Acid SCHEMBL6756464 0.65 HDAC3 (0.38) NPY4RADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326403-B1 CARDIOVASCULAR DISORDERS MERCK PATENT GESELLSCHAFT MIT (DE) 2001-12-04 US claimed
EP-1097127-B1 DIACYLHYDRAZINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2003-03-12 EP disclosed
US-6326403-B1 CARDIOVASCULAR DISORDERS MERCK PATENT GESELLSCHAFT MIT (DE) 2001-12-04 US disclosed