SCHEMBL7879657

SCHEMBL7879657

CN(C(=O)NN[C@@H](CC(=O)O)C(N)=O)C(=O)c1ccccc1NC(=N)N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 4/20 0.39
MAPT P10636 2/20 0.37
KDM4E B2RXH2 4/20 0.36
RECQL P46063 1/20 0.36
ALDH1A1 P00352 3/20 0.35
POLB P06746 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
GAA P10253 1/20 0.34
MASP2 O00187 1/20 0.34
HPGD P15428 2/20 0.33
PRSS1 P07477 1/20 0.33
TMPRSS15 P98073 1/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
LMNA P02545 1/20 0.32
CTSK P43235 1/20 0.32
KMT2A Q03164 1/20 0.32
PYGL P06737 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7878241 0.85 KCNA5 (0.37) ABCC1MAPTKDM4EALDH1A1POLB
SCHEMBL6937428 0.81 ITGB3 (0.40) ITGB3ITGA2BHPGDPRSS1TMPRSS15
SCHEMBL6938684 0.80 ITGB3 (0.43) MAPTALDH1A1ITGB3ITGA2BLMNA
SCHEMBL7878251 0.76 PRSS1 (0.35) ITGB3ITGA2BPRSS1TMPRSS15
SCHEMBL6939377 0.74 SELP (0.36) ITGB3ITGA2B
SCHEMBL6940902 0.74 MEP1B (0.40) ITGB3ITGA2BPRSS1TMPRSS15KMT2A
SCHEMBL6938012 0.68 NPY4R (0.32)
SCHEMBL233797 0.67 KMT2A (0.57) ABCC1MAPTKDM4EALDH1A1POLB
Benzene SCHEMBL27690342 0.67 KMT2A (0.57) ABCC1MAPTKDM4EALDH1A1POLB
Hydrochloric Acid SCHEMBL6013658 0.65 KMT2A (0.55) ABCC1MAPTKDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326403-B1 CARDIOVASCULAR DISORDERS MERCK PATENT GESELLSCHAFT MIT (DE) 2001-12-04 US disclosed