SCHEMBL6941995

SCHEMBL6941995

CN(C)c1ccccc1CC1CCCCC1(O)Cc1c(F)cccc1Cl

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.37
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34
TRPA1 O75762 1/20 0.34
ALDH1A1 P00352 5/20 0.33
LMNA P02545 1/20 0.33
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
SLC6A4 P31645 2/20 0.32
P2RX7 Q99572 1/20 0.32
MAPK1 P28482 1/20 0.32
SLC6A3 Q01959 1/20 0.32
MAPT P10636 2/20 0.32
KDM4E B2RXH2 2/20 0.32
TSHR P16473 2/20 0.32
POLB P06746 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
SLC6A2 P23975 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5846181 0.86 ALDH1A1 (0.38) GAATRPA1ALDH1A1KMT2AMEN1
SCHEMBL6937028 0.86 TRPA1 (0.38) ESR1TRPA1ALDH1A1LMNAKMT2A
SCHEMBL6939503 0.85 TRPA1 (0.36) ESR1GAATRPA1KMT2AMEN1
Hydrochloric Acid SCHEMBL5846854 0.85 ALDH1A1 (0.38) GAATRPA1ALDH1A1KMT2AMEN1
SCHEMBL10451681 0.83 SLC6A4 (0.45) GAAKMT2AMEN1SLC6A4SLC6A3
SCHEMBL10451679 0.83 SLC6A4 (0.45) GAAKMT2AMEN1SLC6A4SLC6A3
SCHEMBL10451711 0.83 SLC6A4 (0.45) GAAKMT2AMEN1SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL10450226 0.82 SLC6A4 (0.44) GAAKMT2AMEN1SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL10451848 0.82 SLC6A4 (0.44) GAAKMT2AMEN1SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL10450224 0.82 SLC6A4 (0.44) GAAKMT2AMEN1SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1043307-B1 3-amino-3-arylpropan-1-ol-derivates, their preparation and their use GRUENENTHAL GMBH (DE) 2003-06-04 EP claimed
US-6410790-B1 ANALGESICS GRUENENTHAL GMBH (DE) 2002-06-25 US claimed
US-6410790-B1 ANALGESICS GRUENENTHAL GMBH (DE) 2002-06-25 US disclosed