SCHEMBL6937028

SCHEMBL6937028

CN(C)c1ccccc1CC1CCCCC1(O)Cc1ccccc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 3/20 0.38
MEN1 O00255 6/20 0.34
KMT2A Q03164 6/20 0.34
ESR1 P03372 1/20 0.34
SLC6A2 P23975 5/20 0.33
SLC6A4 P31645 5/20 0.33
OPRM1 P35372 4/20 0.33
OPRD1 P41143 2/20 0.33
OPRK1 P41145 2/20 0.33
TAAR1 Q96RJ0 1/20 0.33
USP2 O75604 1/20 0.32
TSHR P16473 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
GRIN2B Q13224 1/20 0.32
SLC22A1 O15245 2/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6939503 0.92 TRPA1 (0.36) TRPA1MEN1KMT2AESR1SLC6A2
SCHEMBL6939845 0.90 TRPA1 (0.38) TRPA1MEN1KMT2ASLC6A2SLC6A4
SCHEMBL6937466 0.90 DPP4 (0.35) TRPA1MEN1KMT2ASLC6A2SLC6A4
SCHEMBL6675819 0.88 TAAR1 (0.37) TRPA1MEN1KMT2AESR1SLC6A2
SCHEMBL6937424 0.86 TRPA1 (0.44) TRPA1MEN1KMT2AESR1SLC6A2
SCHEMBL6941995 0.86 ESR1 (0.37) TRPA1MEN1KMT2AESR1SLC6A2
SCHEMBL5846181 0.86 ALDH1A1 (0.38) TRPA1MEN1KMT2ASLC6A2SLC6A4
SCHEMBL5845144 0.85 TRPA1 (0.35) TRPA1MEN1KMT2AESR1SLC6A2
SCHEMBL6936768 0.85 SLC6A9 (0.39) TRPA1MEN1KMT2ASLC6A2SLC6A4
Hydrochloric Acid SCHEMBL5846854 0.85 ALDH1A1 (0.38) TRPA1MEN1KMT2ASLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1043307-B1 3-amino-3-arylpropan-1-ol-derivates, their preparation and their use GRUENENTHAL GMBH (DE) 2003-06-04 EP claimed
US-6410790-B1 ANALGESICS GRUENENTHAL GMBH (DE) 2002-06-25 US claimed
US-6410790-B1 ANALGESICS GRUENENTHAL GMBH (DE) 2002-06-25 US disclosed