SCHEMBL6942591

SCHEMBL6942591

CCCC(C[C@H]([C@H](C/C=C/c1ccccc1)C(=O)NO)[N+]1(C)CCOCC1)(C(=O)NN)S(C)(=O)=O

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 1/20 0.38
CTSC P53634 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA7 P36544 1/20 0.31
CHRNA4 P43681 1/20 0.31
KDM4E B2RXH2 1/20 0.30
USP2 O75604 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
CASP1 P29466 1/20 0.30
CASP7 P55210 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7938335 0.88 TGFBR1 (0.33)
SCHEMBL7100106 0.79 ADAM17 (0.40) ADAM17CHRNB2CHRNB4CHRNA3CHRNA7
Hydrochloric Acid SCHEMBL7105152 0.79 ADAM17 (0.40) ADAM17
SCHEMBL6940773 0.78 ADAM17 (0.40) ADAM17CTSC
SCHEMBL6942646 0.78 ADAM17 (0.40) ADAM17CTSCALDH1A1
SCHEMBL6939564 0.78 ADAM17 (0.40) ADAM17CTSCKDM4E
SCHEMBL6984341 0.77 ADAM17 (0.35) ADAM17
SCHEMBL6944612 0.76 ADAM17 (0.38) ADAM17CTSC
SCHEMBL8111670 0.75 ADAM17 (0.38) ADAM17CTSC
SCHEMBL6944954 0.74 ADAM17 (0.37) ADAM17CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed
EP-0993442-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-04-19 EP disclosed
WO-1999001428-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-01-14 WO disclosed