SCHEMBL6940773

SCHEMBL6940773

C=C(C)C[C@H](CC(CCC)(C(=O)NN)S(C)(=O)=O)[C@H](C/C=C/c1ccccc1)C(=O)NO

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 2/20 0.40
CTSC P53634 1/20 0.33
MASP2 O00187 1/20 0.31
MMP1 P03956 1/20 0.30
MMP9 P14780 1/20 0.30
MMP13 P45452 1/20 0.30
GRIK1 P39086 2/20 0.30
GRIK2 Q13002 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6939564 0.86 ADAM17 (0.40) ADAM17CTSCMASP2MMP13GRIK1
SCHEMBL6946755 0.85 TGFBR1 (0.32)
SCHEMBL6942646 0.81 ADAM17 (0.40) ADAM17CTSCMASP2MMP1MMP9
SCHEMBL6944612 0.79 ADAM17 (0.38) ADAM17CTSC
SCHEMBL6942591 0.78 ADAM17 (0.38) ADAM17CTSC
SCHEMBL8111670 0.78 ADAM17 (0.38) ADAM17CTSC
SCHEMBL6944954 0.78 ADAM17 (0.37) ADAM17CTSCMASP2
SCHEMBL6944604 0.77 ADAM17 (0.36) ADAM17CTSCMASP2MMP1MMP9
SCHEMBL6942160 0.76 ADAM17 (0.37) ADAM17CTSCMASP2MMP1MMP9
SCHEMBL6943076 0.76 ADAM17 (0.39) ADAM17GRIK1GRIK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed