SCHEMBL6943008

SCHEMBL6943008

CCC[C@](C(=O)NN)(c1ccc(C)cc1C(C/C=C/c1cccnc1)C(=O)NO)S(C)(=O)=O

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 17/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
HDAC3 O15379 2/20 0.33
NCOR2 Q9Y618 1/20 0.33
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC11 Q96DB2 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
HDAC9 Q9UKV0 1/20 0.32
HDAC5 Q9UQL6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6942211 0.92 NAMPT (0.35) NAMPTCHRNB2CHRNA4HDAC3NCOR2
SCHEMBL6940940 0.91 ADAM17 (0.35)
SCHEMBL6946167 0.89 NAMPT (0.35) NAMPTCHRNB2CHRNA4
SCHEMBL6943304 0.86 TGFBR1 (0.34) NAMPT
SCHEMBL6944737 0.85 MMP9 (0.36) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL6943877 0.84
SCHEMBL6940117 0.84 GRIK1 (0.35) HDAC1
SCHEMBL6940907 0.82 ADAM17 (0.33)
SCHEMBL6945854 0.82 ADAM17 (0.37)
SCHEMBL6942799 0.81 ADAM17 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed