SCHEMBL6944405

SCHEMBL6944405

Nc1ncc2nc(Cc3ccccn3)[nH]c2n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.48
F10 P00742 1/20 0.48
F7 P08709 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.41
HRH3 Q9Y5N1 2/20 0.39
HRH4 Q9H3N8 1/20 0.39
PDE9A O76083 1/20 0.39
PNP P00491 1/20 0.38
ASIC3 Q9UHC3 1/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPT P10636 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP2E1 P05181 2/20 0.36
CYP2C8 P10632 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31595169 0.78 F2 (0.48) F2F10F7L3MBTL1HRH3
SCHEMBL6946589 0.77 MAPT (0.37) HRH3HRH4MAPTKDM4ECYP1A2
SCHEMBL6945088 0.74 CYP1A2 (0.48) MAPTMEN1KMT2ACYP1A2CYP2D6
SCHEMBL6950878 0.74 RAB9A (0.53) ALDH1A1MAPTHTTLMNASMN1; SMN2
SCHEMBL3338581 0.73 F2 (0.61) F2F10F7CYP1A2CYP2E1
SCHEMBL6947942 0.73 EGFR (0.43) MAPTKDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL6948071 0.72 RAB9A (0.44) ALDH1A1MAPTCYP2D6SMN1; SMN2POLB
SCHEMBL6946765 0.72 CYP2D6 (0.44) ALDH1A1MAPTCYP2D6MAOBSMN1; SMN2
SCHEMBL6939915 0.72 DHFR (0.56) MAPTKDM4EKMT2ACYP1A2CYP3A4
SCHEMBL6948821 0.72 MAPT (0.40) L3MBTL1ALDH1A1MAPTCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed