SCHEMBL6944407

SCHEMBL6944407

Nc1ncc2ncn(Cc3ccccn3)c2n1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.50
HSP90AA1 P07900 1/20 0.46
HSP90AB1 P08238 1/20 0.46
SLC29A1 Q99808 2/20 0.45
SLC2A1 P11166 1/20 0.44
CYP1A2 P05177 1/20 0.44
LMNA P02545 1/20 0.43
TLR7 Q9NYK1 10/20 0.42
HTR2A P28223 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
ADRA1A P35348 1/20 0.41
HSD17B10 Q99714 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
KCNH2 Q12809 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28299548 0.81 HDAC6 (0.63) HDAC6HSP90AA1HSP90AB1CYP1A2KDM4E
SCHEMBL6343841 0.81 ADRA1D (0.44) HDAC6SLC2A1LMNAKDM4EALDH1A1
SCHEMBL6946592 0.77 HDAC6 (0.62) HDAC6HSP90AA1HSP90AB1CYP1A2TLR7
SCHEMBL6944465 0.77 HDAC6 (0.55) HDAC6HSP90AA1HSP90AB1CYP1A2LMNA
SCHEMBL11146983 0.75 ALDH1A1 (0.46) SLC2A1LMNATLR7KDM4EALDH1A1
SCHEMBL4961031 0.75 HDAC6 (0.52) HDAC6HSP90AA1HSP90AB1CYP1A2KDM4E
SCHEMBL6945092 0.73 HDAC6 (0.64) HDAC6HSP90AA1HSP90AB1CYP1A2LMNA
SCHEMBL6950880 0.73 HTT (0.54) HDAC6HSP90AA1HSP90AB1CYP1A2LMNA
SCHEMBL14642669 0.72 CDK1 (0.56) HDAC6HSP90AA1HSP90AB1SLC29A1TLR7
SCHEMBL6947944 0.72 ALDH1A1 (0.56) HDAC6HSP90AA1HSP90AB1SLC2A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed