SCHEMBL6944455

SCHEMBL6944455

Nc1nc(Cc2cccnc2)c2nc[nH]c2n1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 3/20 0.44
HRH3 Q9Y5N1 3/20 0.44
PNP P00491 1/20 0.41
MPO P05164 2/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MGMT P16455 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2D6 P10635 1/20 0.37
MMP2 P08253 1/20 0.37
CHRNA7 P36544 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
NAMPT P43490 1/20 0.36
CYP3A4 P08684 1/20 0.36
DHFR P00374 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10435291 0.84 HRH4 (0.44) HRH4HRH3PNPMPOKMT2A
SCHEMBL6946585 0.83 MPO (0.40) HRH4HRH3PNPMPOMGMT
SCHEMBL6939911 0.78 DHFR (0.47) MPOKMT2AMGMTCYP1A2CYP2D6
SCHEMBL6947940 0.78 PIN1 (0.48) HRH4MPO
SCHEMBL6945083 0.77 PIN1 (0.44) MPOCYP1A2CYP2D6CYP3A4DHFR
SCHEMBL6948619 0.76 PNP (0.41) PNPMPO
SCHEMBL6944400 0.76 HRH3 (0.42) HRH4HRH3PNPMPOMGMT
SCHEMBL6948069 0.76 MPO (0.47) HRH3MPOMGMTCYP1A2CYP2D6
SCHEMBL6946759 0.76 CYP2D6 (0.48) HRH3MPOCYP1A2CYP2D6CYP3A4
SCHEMBL6950876 0.75 MPO (0.56) MPOMGMTCYP1A2CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed