SCHEMBL6946585

SCHEMBL6946585

Nc1nc(Cc2ccncc2)c2nc[nH]c2n1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.40
HRH4 Q9H3N8 2/20 0.38
HRH3 Q9Y5N1 2/20 0.38
CYP3A4 P08684 3/20 0.37
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PNP P00491 1/20 0.36
CYP17A1 P05093 4/20 0.36
CYP11B1 P15538 4/20 0.36
CYP11B2 P19099 4/20 0.36
CYP19A1 P11511 3/20 0.36
HTR6 P50406 1/20 0.34
MGMT P16455 3/20 0.33
CDK1 P06493 1/20 0.32
RAB9A P51151 1/20 0.32
LOXL2 Q9Y4K0 1/20 0.32
ADORA2A P29274 1/20 0.31
FLT1 P17948 3/20 0.31
KDR P35968 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6945083 0.84 PIN1 (0.44) MPOCYP3A4SMN1; SMN2HTR6KDR
SCHEMBL6944455 0.83 HRH4 (0.44) MPOHRH4HRH3CYP3A4PNP
SCHEMBL10435362 0.82 HRH4 (0.38) HRH4HRH3CYP3A4MAPTSMN1; SMN2
SCHEMBL6941905 0.81 ALDH1A1 (0.50) MPOMAPTSMN1; SMN2HTR6
SCHEMBL6948619 0.80 PNP (0.41) MPOPNPCDK1ADORA2A
SCHEMBL6944400 0.77 HRH3 (0.42) MPOHRH4HRH3PNPMGMT
SCHEMBL6947940 0.77 PIN1 (0.48) MPOHRH4HTR6RAB9AADORA2A
SCHEMBL6939911 0.77 DHFR (0.47) MPOCYP3A4MAPTMGMTCDK1
SCHEMBL6950768 0.76 CYP17A1 (0.39) MPOCYP3A4CYP17A1CYP11B1CYP11B2
Ammonia Solution, Strong SCHEMBL17009431 0.75 KDM4A (0.41) MPOSMN1; SMN2PNPMGMTADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed