SCHEMBL6944895

SCHEMBL6944895

CN(C)CC1CC(Cc2ccc(Cl)cc2)CCC1(O)C#C[Si](C)(C)C.COc1ccc(C2(O)CCC(Cc3ccc(Cl)cc3)CC2CN(C)C)cc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 7/20 0.37
OPRM1 P35372 5/20 0.36
OPRD1 P41143 4/20 0.36
SLC6A2 P23975 4/20 0.36
SLC6A4 P31645 4/20 0.36
SLC22A1 O15245 2/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
AVPR1A P37288 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
EDNRA P25101 1/20 0.33
SCN9A Q15858 1/20 0.31
SLC6A9 P48067 1/20 0.31
SLC6A5 Q9Y345 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4665474 0.89 OPRK1 (0.43) OPRK1OPRM1OPRD1SLC6A2SLC6A4
SCHEMBL4663384 0.88 OPRM1 (0.33) OPRK1OPRM1OPRD1SLC6A4ALDH1A1
SCHEMBL4665379 0.82 OPRK1 (0.42) OPRK1OPRM1OPRD1SLC6A2SLC6A4
SCHEMBL4663457 0.80 OPRM1 (0.43) OPRK1OPRM1OPRD1SLC6A2SLC6A4
SCHEMBL4665371 0.78 OPRK1 (0.39) OPRK1OPRM1OPRD1SLC6A2SLC6A4
SCHEMBL4663680 0.78 OPRK1 (0.60) OPRK1OPRM1OPRD1SLC6A2SLC6A4
SCHEMBL4663394 0.78 OPRK1 (0.53) OPRK1OPRM1OPRD1SLC6A2SLC6A4
SCHEMBL4665354 0.77 DRD2 (0.41) OPRK1OPRM1OPRD1SLC6A2SLC6A4
SCHEMBL4663483 0.77 DRD2 (0.41) OPRK1OPRM1OPRD1SLC6A2SLC6A4
SCHEMBL4664046 0.77 SMN1; SMN2 (0.48) OPRK1OPRM1OPRD1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368299-A2 SUBSTITUTED C-CYCLOHEXYLMETHYLAMINE DERIVATIVES Grünenthal GmbH (DE) 2003-12-10 EP disclosed
WO-2002030870-A2 SUBSTITUTED C-CYCLOHEXYLMETHYLAMINE DERIVATIVES Grünenthal GmbH (DE) 2002-04-18 WO disclosed