SCHEMBL6945304

SCHEMBL6945304

CCOCOc1ccc(-c2cc(OCOCC)ccc2C(=O)c2ccc(OCCC3CCCCN3)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.49
HCRTR1 O43613 1/20 0.43
HCRTR2 O43614 1/20 0.43
SSTR2 P30874 7/20 0.41
LTA4H P09960 3/20 0.41
CNR2 P34972 2/20 0.38
PRKAB2 O43741 1/20 0.37
PRKAG1 P54619 1/20 0.37
PRKAA2 P54646 1/20 0.37
PRKAA1 Q13131 1/20 0.37
PRKAG3 Q9UGI9 1/20 0.37
PRKAG2 Q9UGJ0 1/20 0.37
PRKAB1 Q9Y478 1/20 0.37
AURKB Q96GD4 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
RECQL P46063 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6765314 0.75 CHEK2 (0.52) CHEK2MAPTHRH2HRH1
SCHEMBL8716635 0.75 CHEK2 (0.46) CHEK2HCRTR1HCRTR2LTA4HKDM4E
SCHEMBL6053346 0.75 CHEK2 (0.58) CHEK2LTA4HHRH2HRH1
SCHEMBL7335065 0.75 LTA4H (0.54) CHEK2LTA4HKDM4EALDH1A1
SCHEMBL7447377 0.74 LTA4H (0.56) CHEK2LTA4HAURKBHRH2HRH1
Hydrochloric Acid SCHEMBL7328923 0.74 LTA4H (0.53) CHEK2LTA4HKDM4EALDH1A1
SCHEMBL11713224 0.73 CHEK2 (0.55) CHEK2SSTR2LTA4HAURKBHRH2
SCHEMBL3866051 0.73 CHEK2 (0.56) CHEK2LTA4HHRH2HRH1
Hydrochloric Acid SCHEMBL7435059 0.73 LTA4H (0.55) CHEK2LTA4HHRH2HRH1
SCHEMBL6560708 0.72 MAPT (0.56) CHEK2LTA4HKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025098-A4 BENZOTHIOPHENES LILLY CO ELI (US) 2003-03-05 EP disclosed
EP-1025098-A1 BENZOTHIOPHENES ELI LILLY AND COMPANY (US) 2000-08-09 EP disclosed
WO-1999018101-A1 BENZOTHIOPHENES ELI LILLY AND COMPANY (US) 1999-04-15 WO disclosed