SCHEMBL6945772

SCHEMBL6945772

COCCOC(=O)C1=C(C)NC(C)=C(C(=O)O)C1c1c(F)cccc1Cl

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.68
TP53 P04637 2/20 0.48
CACNA1B Q00975 5/20 0.48
CYP2C9 P11712 5/20 0.47
CYP1A2 P05177 4/20 0.47
CYP3A4 P08684 4/20 0.47
CYP2C19 P33261 4/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
KDM4E B2RXH2 2/20 0.47
HIF1A Q16665 2/20 0.47
HSD17B10 Q99714 2/20 0.47
MAPT P10636 2/20 0.47
MTOR P42345 2/20 0.47
CYP2D6 P10635 2/20 0.47
TSHR P16473 2/20 0.47
NFKB1 P19838 2/20 0.47
THPO P40225 2/20 0.47
LMNA P02545 2/20 0.47
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947853 0.92 ALOX15 (0.59) ALOX15CACNA1BCYP2C9CYP1A2CYP3A4
SCHEMBL6944706 0.89 ALOX15 (0.64) ALOX15TP53CYP2C9CYP1A2CYP3A4
SCHEMBL6950055 0.86 POLB (0.49) ALOX15TP53CACNA1BCYP2C9CYP1A2
SCHEMBL6949599 0.86 ALOX15 (0.61) ALOX15TP53CYP2C9CYP1A2CYP3A4
SCHEMBL6952565 0.83 ALOX15 (0.61) ALOX15TP53CYP2C9CYP1A2CYP3A4
SCHEMBL6945817 0.82 ALOX15 (0.51) ALOX15TP53CACNA1BCYP2C9CYP1A2
SCHEMBL7275334 0.82 CYP2C9 (0.70) ALOX15TP53CACNA1BCYP2C9CYP1A2
SCHEMBL7267278 0.82 CYP2C9 (0.57) ALOX15TP53CACNA1BCYP2C9CYP1A2
SCHEMBL6950016 0.82 ALOX15 (0.50) ALOX15CACNA1BKDM4EMAPTALDH1A1
SCHEMBL9246654 0.81 MAPT (0.62) ALOX15TP53CYP2C9CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657432-B1 Phenyl-substituted 1,4-dihydropyridines with cerebral activity BAYER AG (DE) 2003-03-12 EP claimed