SCHEMBL6946474

SCHEMBL6946474

O=C1c2ccccc2C(=O)N1CC(CCO)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 2/20 0.49
RAB9A P51151 1/20 0.42
ALDH1A1 P00352 3/20 0.40
ALOX15 P16050 2/20 0.39
HSD17B10 Q99714 2/20 0.39
APAF1 O14727 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
BCHE P06276 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
ALOX12 P18054 1/20 0.39
ACHE P22303 1/20 0.39
CES1 P23141 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6604494 0.82 TNF (0.46) TNFRAB9AALDH1A1ALOX15HSD17B10
SCHEMBL6604487 0.82 TNF (0.46) TNFRAB9AALDH1A1ALOX15HSD17B10
SCHEMBL3912571 0.70 SLC6A2 (0.43) ALDH1A1CYP1A2CYP3A4CYP2D6MAPT
SCHEMBL4675885 0.70 SLC6A2 (0.43) ALDH1A1CYP1A2CYP3A4CYP2D6MAPT
SCHEMBL8592939 0.70 SLC6A3 (0.38) ALDH1A1CYP3A4CYP2D6HTT
SCHEMBL4712246 0.70 MAPK1 (0.55) RAB9AALDH1A1MAPTKMT2ACASP3
SCHEMBL8913116 0.70 PRKCZ (0.49) ALDH1A1CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL18756303 0.69 LTA4H (0.51) RAB9AALDH1A1MAPTKMT2ACASP3
SCHEMBL18222526 0.69 ALDH1A1 (0.49) TNFRAB9AALDH1A1MAPTKMT2A
SCHEMBL7260089 0.69 ALDH1A1 (0.49) TNFRAB9AALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709376-B1 Phenylpiperidino derivatives as neurokinin antagonists ASTRAZENECA AB (SE) 2003-07-23 EP disclosed
US-6008223-A ANTIINFLAMMATORY AGENTS FOR TREATING ASTHMA ZENECA LIMITED (GB) 1999-12-28 US disclosed
US-5731309-A Substituted heteroalkyleneamine neurokinin antagonists ZENECA LIMITED (GB) 1998-03-24 US disclosed
EP-0709376-A2 Therapeutic compounds ZENECA LIMITED (GB) 1996-05-01 EP disclosed