SCHEMBL6948194

SCHEMBL6948194

Nc1ncc2ncn(Cc3cccc4[nH]ccc34)c2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.45
HSP90AB1 P08238 1/20 0.45
HDAC6 Q9UBN7 2/20 0.44
ADORA2A P29274 6/20 0.41
DAO P14920 1/20 0.39
HTT P42858 1/20 0.38
HCRTR1 O43613 3/20 0.37
HCRTR2 O43614 3/20 0.37
ADORA1 P30542 3/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
ADRA1A P35348 1/20 0.36
HSD17B10 Q99714 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
DHFR P00374 1/20 0.34
PIK3CA P42336 1/20 0.33
MTOR P42345 1/20 0.33
PDE2A O00408 1/20 0.33
MET P08581 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950775 0.75 HDAC6 (0.53) HSP90AA1HSP90AB1HDAC6ADORA2AADORA1
SCHEMBL3269002 0.75 ADORA2A (0.75) ADORA2AADORA1
SCHEMBL28299548 0.72 HDAC6 (0.63) HSP90AA1HSP90AB1HDAC6ADORA2AADORA1
SCHEMBL6948823 0.71 HDAC6 (0.47) HSP90AA1HSP90AB1HDAC6ADORA2AHTT
SCHEMBL6948190 0.71 KRAS (0.40) DAOHTTDHFRPIK3CAMTOR
SCHEMBL6944407 0.69 HDAC6 (0.50) HSP90AA1HSP90AB1HDAC6KDM4EALDH1A1
SCHEMBL4961031 0.69 HDAC6 (0.52) HSP90AA1HSP90AB1HDAC6ADORA2AADORA1
SCHEMBL6939917 0.68 HDAC6 (0.56) HSP90AA1HSP90AB1HDAC6ADORA2AADORA1
SCHEMBL6947944 0.68 ALDH1A1 (0.56) HSP90AA1HSP90AB1HDAC6ADORA2AHTT
SCHEMBL29761060 0.68 HDAC6 (0.67) HSP90AA1HSP90AB1HDAC6ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed