SCHEMBL6948942

SCHEMBL6948942

COC(=O)CC(=O)c1cccc2[nH]c(CCc3ccccc3)nc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.50
CREBBP Q92793 1/20 0.50
PARP1 P09874 2/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
MMP2 P08253 1/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NTRK1 P04629 3/20 0.43
HDAC6 Q9UBN7 1/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
RIPK1 Q13546 1/20 0.42
GAA P10253 1/20 0.41
DHODH Q02127 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6949839 0.90 CHEK1 (0.50) BRD4CREBBPPARP1NPC1RAB9A
SCHEMBL6946441 0.89 PARP1 (0.48) BRD4CREBBPPARP1NPC1RAB9A
SCHEMBL6946473 0.88 NPC1 (0.50) BRD4CREBBPPARP1NPC1RAB9A
SCHEMBL6948419 0.85 PARP1 (0.45) BRD4CREBBPPARP1NPC1RAB9A
SCHEMBL6945364 0.83 RAB9A (0.52) BRD4CREBBPPARP1NPC1RAB9A
SCHEMBL6948954 0.82 NPC1 (0.55) PARP1NPC1RAB9AKDM4EHDAC6
SCHEMBL6948273 0.82 DHODH (0.51) BRD4CREBBPPARP1ALDH1A1MAPT
SCHEMBL6945300 0.81 CHEK1 (0.48) BRD4CREBBPPARP1MAPTHSD17B10
SCHEMBL6948946 0.81 NPC1 (0.46) BRD4CREBBPPARP1NPC1RAB9A
SCHEMBL29412049 0.80 PARP1 (0.60) PARP1NPC1RAB9ADHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0936218-B1 BENZIMIDAZOLE DERIVATIVES MOCHIDA PHARM CO LTD (JP) 2003-04-02 EP disclosed
US-6387938-B1 Benzimidazole derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2002-05-14 US disclosed
EP-0936218-A1 NOVEL BENZIMIDAZOLE DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1999-08-18 EP disclosed