SCHEMBL6949388

SCHEMBL6949388

COc1c(Br)cc(Cc2ccccc2)cc1N(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.42
NQO2 P16083 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
MAPT P10636 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
THRB P10828 2/20 0.38
KDM4E B2RXH2 2/20 0.38
GAA P10253 2/20 0.38
ALDH1A1 P00352 1/20 0.38
BLM P54132 1/20 0.38
HTT P42858 1/20 0.36
CALM1 P0DP23 1/20 0.36
POLB P06746 1/20 0.35
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946183 0.85 LTA4H (0.52) LTA4HNQO2SMN1; SMN2LMNAHPGD
SCHEMBL6947814 0.80 LMNA (0.53) LTA4HSMN1; SMN2LMNAHPGDMAPT
SCHEMBL6949776 0.79 ALDH1A1 (0.41) LTA4HSMN1; SMN2LMNAHPGDMEN1
SCHEMBL6950237 0.78 LTA4H (0.44) LTA4HNQO2SMN1; SMN2LMNAHPGD
SCHEMBL6943711 0.77 LTA4H (0.43) LTA4HSMN1; SMN2LMNAHPGDMAPT
SCHEMBL7077380 0.76 LTA4H (0.42) LTA4HSMN1; SMN2LMNAHPGDMAPT
SCHEMBL6946931 0.72 LMNA (0.41) LTA4HSMN1; SMN2LMNAHPGDMAPT
SCHEMBL6947888 0.72 ERCC5 (0.42) ALDH1A1
SCHEMBL6950123 0.71 KMT2A (0.49) LTA4HSMN1; SMN2LMNAHPGDMAPT
SCHEMBL6946141 0.70 KMT2A (0.49) SMN1; SMN2LMNAHPGDMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed