SCHEMBL6950237

SCHEMBL6950237

COc1c(N)cc(Cc2ccccc2)cc1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.44
GAA P10253 2/20 0.42
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CALM1 P0DP23 1/20 0.39
ALDH1A1 P00352 2/20 0.39
NQO2 P16083 1/20 0.37
MAPT P10636 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
THRB P10828 2/20 0.37
KDM4E B2RXH2 1/20 0.37
BLM P54132 1/20 0.37
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946183 0.88 LTA4H (0.52) LTA4HGAALMNAHPGDSMN1; SMN2
SCHEMBL6947814 0.82 LMNA (0.53) LTA4HGAALMNAHPGDSMN1; SMN2
SCHEMBL6943711 0.79 LTA4H (0.43) LTA4HLMNAHPGDSMN1; SMN2CALM1
SCHEMBL6949388 0.78 LTA4H (0.42) LTA4HGAALMNAHPGDSMN1; SMN2
SCHEMBL7077380 0.78 LTA4H (0.42) LTA4HLMNAHPGDSMN1; SMN2CALM1
SCHEMBL30079648 0.76 CA2 (0.39) GAAALDH1A1MAPTMEN1KMT2A
SCHEMBL27171654 0.76 CA2 (0.39) GAAALDH1A1MAPTMEN1KMT2A
SCHEMBL6949776 0.76 ALDH1A1 (0.41) LTA4HLMNAHPGDSMN1; SMN2ALDH1A1
SCHEMBL6946931 0.75 LMNA (0.41) LTA4HGAALMNAHPGDSMN1; SMN2
SCHEMBL6948033 0.75 PTPN1 (0.47) LMNAHPGDCALM1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed