SCHEMBL6949402

SCHEMBL6949402

COC(=O)c1ccc(C2C(O)CN(OC(=O)OC(C)(C)C)CC2CO)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HSD17B10 Q99714 3/20 0.34
ALDH1A1 P00352 3/20 0.34
TSHR P16473 2/20 0.34
KDM4E B2RXH2 2/20 0.34
GAA P10253 2/20 0.34
HPGD P15428 2/20 0.34
CASP1 P29466 2/20 0.34
CASP7 P55210 2/20 0.34
ATM Q13315 2/20 0.34
GRM2 Q14416 1/20 0.34
HTT P42858 2/20 0.33
RAB9A P51151 2/20 0.33
PDE4B Q07343 1/20 0.33
NPC1 O15118 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPK1 P28482 1/20 0.32
GLA P06280 1/20 0.32
MEN1 O00255 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1942520 0.87 PDE4B (0.33) PDE4B
SCHEMBL6948019 0.86 RORC (0.36) ALDH1A1GAAHTTRAB9APDE4B
SCHEMBL6959407 0.84 HDAC1 (0.34) HDAC1HDAC6HSD17B10ALDH1A1TSHR
SCHEMBL2254270 0.83 PDE4B (0.46) HDAC1HDAC6KDM4EPDE4BKMT2A
SCHEMBL6953398 0.80 PDE4B (0.35) PDE4B
SCHEMBL6960005 0.78 MEN1 (0.39) HDAC1HDAC6HSD17B10ALDH1A1TSHR
SCHEMBL6042971 0.77 ALDH1A1 (0.39) HSD17B10ALDH1A1TSHRKDM4EGAA
SCHEMBL6955257 0.76 MIF (0.35) PDE4B
SCHEMBL6951399 0.76 SLC6A3 (0.37) ALDH1A1KMT2A
SCHEMBL6955012 0.75 REN (0.41) ALDH1A1KDM4EPDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863875-B1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY HOFFMANN LA ROCHE (CH) 2003-06-04 EP disclosed
EP-0863875-A1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY F. HOFFMANN-LA ROCHE AG (CH) 1998-09-16 EP disclosed
WO-1997009311-A1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY F. HOFFMANN-LA ROCHE AG (CH) 1997-03-13 WO disclosed