SCHEMBL6953191

SCHEMBL6953191

Nc1cccc(COC(=O)c2ccccc2C=O)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
TDP1 Q9NUW8 4/20 0.46
RAB9A P51151 3/20 0.43
KDM4E B2RXH2 2/20 0.43
GAA P10253 1/20 0.43
STAT1 P42224 1/20 0.43
POLB P06746 1/20 0.43
TSHR P16473 3/20 0.41
CYP3A4 P08684 2/20 0.41
MAPK1 P28482 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
KMT2A Q03164 3/20 0.40
HPGD P15428 2/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
GLA P06280 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HIF1A Q16665 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL381019 0.84 ALDH1A1 (0.65) ALDH1A1TDP1RAB9APOLBTSHR
SCHEMBL18625926 0.79 TDP1 (0.55) ALDH1A1TDP1RAB9AKDM4EPOLB
SCHEMBL7351514 0.76 ALDH1A1 (0.48) ALDH1A1TDP1RAB9AKDM4EGAA
SCHEMBL28367951 0.76 TDP1 (0.60) ALDH1A1TDP1RAB9AKDM4EGAA
SCHEMBL31620922 0.76 MAOB (0.50) ALDH1A1TDP1MAPK1L3MBTL1KMT2A
SCHEMBL1900241 0.74 TDP1 (0.50) ALDH1A1TDP1RAB9AKDM4EGAA
SCHEMBL11403328 0.74 RAB9A (0.56) ALDH1A1TDP1RAB9AKDM4ETSHR
SCHEMBL29878507 0.73 TDP1 (0.56) ALDH1A1TDP1RAB9APOLBTSHR
SCHEMBL6322994 0.73 ALDH1A1 (0.50) ALDH1A1TDP1RAB9APOLBTSHR
SCHEMBL3881721 0.73 THRA (0.47) ALDH1A1TDP1POLBTHRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0758327-B1 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS UPJOHN CO (US) 2003-04-09 EP disclosed
US-6169181-B1 HUMAN IMMUNODEFICIENCY VIRUS PROTEINASE INHIBITORS PHARMACIA & UPJOHN COMPANY 2001-01-02 US disclosed
US-5852195-A Pyranone compounds useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1998-12-22 US disclosed
EP-0758327-A1 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1997-02-19 EP disclosed
WO-1995030670-A2 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-16 WO disclosed