SCHEMBL6953405

SCHEMBL6953405

NC(=O)COc1ccc2c(C(=O)O)c(CN3CCCC(C4CCNCC4)C3)c(-c3ccccc3)nc2c1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 8/20 0.41
TACR2 P21452 7/20 0.41
OPRM1 P35372 4/20 0.41
KCNH2 Q12809 2/20 0.39
TRPV4 Q9HBA0 4/20 0.38
NR1I2 O75469 1/20 0.38
ROCK2 O75116 1/20 0.37
ACACA Q13085 1/20 0.36
CHEK2 O96017 2/20 0.36
DPP4 P27487 2/20 0.36
LCK P06239 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6957439 0.86 TACR3 (0.46) TACR3TACR2OPRM1KCNH2TRPV4
SCHEMBL6957829 0.85 TACR3 (0.54) TACR3TACR2OPRM1KCNH2TRPV4
Hydrochloric Acid SCHEMBL6958335 0.84 TACR3 (0.53) TACR3TACR2OPRM1KCNH2TRPV4
Hydrochloric Acid SCHEMBL6953706 0.81 TACR3 (0.41) TACR3TACR2OPRM1KCNH2TRPV4
SCHEMBL5945414 0.80 TRPV4 (0.55) TACR3TACR2OPRM1TRPV4NR1I2
SCHEMBL6959275 0.79 TACR3 (0.55) TACR3TACR2OPRM1KCNH2TRPV4
SCHEMBL6950894 0.79 TACR3 (0.40) TACR3TACR2OPRM1KCNH2TRPV4
SCHEMBL6626342 0.78 TRPV4 (0.50) TACR3TACR2OPRM1KCNH2TRPV4
Bromide SCHEMBL6948962 0.76 TACR3 (0.39) TACR3TACR2OPRM1KCNH2TRPV4
SCHEMBL6627408 0.75 TACR3 (0.43) TACR3TACR2OPRM1KCNH2TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339691-A1 NOVEL COMPOUNDS GlaxoSmithKline S.p.A. (IT) 2003-09-03 EP disclosed
WO-2002044154-A1 NOVEL COMPOUNDS GLAXOSMITHKLINE SPA (IT) 2002-06-06 WO disclosed