SCHEMBL6950894

SCHEMBL6950894

CCOC(=O)COc1ccc2c(C(=O)NCCCc3ccccc3)c(CN3CCC[C@@H](C4CCNCC4)C3)c(-c3ccccc3)nc2c1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 7/20 0.40
TACR2 P21452 5/20 0.40
OPRM1 P35372 3/20 0.40
TRPV4 Q9HBA0 3/20 0.40
NR1I2 O75469 1/20 0.40
LMNA P02545 1/20 0.39
ROCK2 O75116 1/20 0.39
KCNH2 Q12809 3/20 0.38
TLR7 Q9NYK1 3/20 0.38
MAPT P10636 1/20 0.37
NAMPT P43490 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6953706 0.92 TACR3 (0.41) TACR3TACR2OPRM1TRPV4NR1I2
SCHEMBL6953405 0.79 TACR3 (0.41) TACR3TACR2OPRM1TRPV4NR1I2
SCHEMBL6959275 0.74 TACR3 (0.55) TACR3TACR2OPRM1TRPV4KCNH2
SCHEMBL6957439 0.72 TACR3 (0.46) TACR3TACR2OPRM1TRPV4KCNH2
SCHEMBL6957829 0.72 TACR3 (0.54) TACR3TACR2OPRM1TRPV4KCNH2
Hydrochloric Acid SCHEMBL6958335 0.71 TACR3 (0.53) TACR3TACR2OPRM1TRPV4KCNH2
SCHEMBL5945384 0.70 TACR3 (0.74) TACR3TACR2OPRM1TRPV4NR1I2
SCHEMBL6626342 0.66 TRPV4 (0.50) TACR3TACR2OPRM1TRPV4KCNH2
Bromide SCHEMBL6948962 0.64 TACR3 (0.39) TACR3TACR2OPRM1TRPV4KCNH2
SCHEMBL7200846 0.64 LMNA (0.52) TACR3TACR2OPRM1TRPV4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339691-A1 NOVEL COMPOUNDS GlaxoSmithKline S.p.A. (IT) 2003-09-03 EP disclosed
WO-2002044154-A1 NOVEL COMPOUNDS GLAXOSMITHKLINE SPA (IT) 2002-06-06 WO disclosed