SCHEMBL6953502

SCHEMBL6953502

O=C1c2ccc([N+](=O)[O-])cc2C(=O)N1CCc1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.71
CA1 P00915 1/20 0.71
CA2 P00918 1/20 0.71
CA4 P22748 1/20 0.71
CA9 Q16790 1/20 0.71
ACHE P22303 3/20 0.61
CASP3 P42574 2/20 0.56
KDM4E B2RXH2 1/20 0.56
CASP1 P29466 1/20 0.55
CASP4 P49662 1/20 0.55
CASP7 P55210 1/20 0.55
CASP9 P55211 1/20 0.55
CASP6 P55212 1/20 0.55
CASP8 Q14790 1/20 0.55
ALOX5 P09917 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21176664 0.86 CA12 (0.70) CA12CA1CA2CA9ACHE
SCHEMBL17550101 0.85 CA1 (0.62) CA12CA1CA2CA4CA9
SCHEMBL29531485 0.85 CA1 (0.62) CA12CA1CA2CA4CA9
SCHEMBL3061314 0.84 ALDH1A1 (0.59) CA12CA1CA2CA4CA9
SCHEMBL5024423 0.80 NPC1 (0.65) CA12CA1CA2CA4CA9
SCHEMBL3586091 0.80 POLB (0.62) CA12CA1CA2CA4CA9
SCHEMBL8090142 0.80 ACHE (0.62) CA12CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL9370152 0.80 ACHE (0.66) ACHE
SCHEMBL4234495 0.79 RAB9A (0.66) CA12CA1CA2CA4CA9
SCHEMBL10462357 0.79 MAOB (0.70) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674623-B1 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2003-04-09 EP disclosed
EP-0593603-B1 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-11-20 EP disclosed
US-6403578-B1 ANTICOAGULANTS, CARDIOVASCULAR DISORDERS SMITHKLINE BEECHAM CORPORATION 2002-06-11 US disclosed
US-6127359-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 2000-10-03 US disclosed
US-5939412-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 1999-08-17 US disclosed
US-5693636-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 1997-12-02 US disclosed
EP-0593603-A1 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1994-04-27 EP disclosed
WO-1993000095-A2 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1993-01-07 WO disclosed