SCHEMBL6954396

SCHEMBL6954396

CCOc1ccc2[nH]cc(CCCCN3CCCC(Cc4ccccc4)C3)c2c1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 3/20 0.50
HTR1B P28222 3/20 0.50
HTR1A P08908 4/20 0.49
ADRA2A P08913 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
ADRA1D P25100 1/20 0.49
ADRA1A P35348 1/20 0.49
ADRA1B P35368 1/20 0.49
SLC6A4 P31645 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960163 0.93 CARM1 (0.45) HTR1DHTR1BHTR1ASLC6A4
SCHEMBL6954556 0.91 HTR1A (0.60) HTR1BHTR1AADRA2AADRA2BADRA2C
SCHEMBL7356374 0.87 HTR1A (0.51) HTR1DHTR1BHTR1ASLC6A4
SCHEMBL7291647 0.87 HTR1A (0.51) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL7358948 0.87 HTR1A (0.54) HTR1DHTR1BHTR1ASLC6A4
SCHEMBL6958383 0.86 HTR1A (0.52) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL6957729 0.85 MPO (0.61) HTR1DHTR1BHTR1AADRA1ASLC6A4
SCHEMBL6958552 0.85 MPO (0.61) HTR1DHTR1BHTR1AADRA1ASLC6A4
SCHEMBL6951363 0.85 HTR1A (0.55) HTR1DHTR1BHTR1ASLC6A4
SCHEMBL6952634 0.85 MPO (0.61) HTR1DHTR1BHTR1AADRA1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993458-B1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 2003-04-09 EP disclosed
US-6333339-B1 CENTRAL SYSTEM DISORDERS, SCHIZOPHRENIA AND COGNITION ACTIVATORS MERCK PATENT GELLSCHAFT MIT BESCHRANKTER (DE) 2001-12-25 US disclosed
EP-0993458-A1 3-BENZYLPIPERIDINE MERCK PATENT GmbH (DE) 2000-04-19 EP disclosed
WO-1998057953-A1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 1998-12-23 WO disclosed