SCHEMBL6966490

SCHEMBL6966490

COc1cc(C)c(C(C)O)cc1NC(=S)N1CCN(c2cc(C)cc(C)c2)CC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.48
MEN1 O00255 4/20 0.48
CYP3A4 P08684 2/20 0.48
POLB P06746 2/20 0.48
CYP2C19 P33261 1/20 0.48
PHGDH O43175 3/20 0.47
PKM P14618 1/20 0.47
RAB9A P51151 1/20 0.45
DUSP3 P51452 1/20 0.45
PTPN11 Q06124 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6963684 0.91 MEN1 (0.55) KMT2AMEN1CYP3A4POLBCYP2C19
SCHEMBL6955540 0.90 PHGDH (0.49) KMT2AMEN1CYP3A4POLBCYP2C19
SCHEMBL6786898 0.88 CYP3A4 (0.55) KMT2AMEN1CYP3A4POLBCYP2C19
SCHEMBL6960712 0.87 RBP4 (0.47) KMT2AMEN1POLBRAB9AALDH1A1
SCHEMBL6966126 0.81 PHGDH (0.51) KMT2AMEN1CYP3A4POLBCYP2C19
SCHEMBL6959643 0.81 MAPT (0.51) KMT2AMEN1CYP3A4POLBCYP2C19
SCHEMBL6965253 0.78 RBP4 (0.49) KMT2APOLBALDH1A1LMNAGAA
SCHEMBL6782760 0.78 CYP3A4 (0.66) KMT2AMEN1CYP3A4POLBCYP2C19
SCHEMBL6783848 0.78 KMT2A (0.63) KMT2AMEN1CYP3A4POLBCYP2C19
SCHEMBL6960488 0.77 PHGDH (0.55) KMT2AMEN1CYP3A4POLBCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850222-B1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARM CO LTD (KR) 2003-05-28 EP disclosed
US-6028195-A AN ANTITUMOR AGENT WITH VERY LOW TOXICITIES SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2000-02-22 US disclosed