SCHEMBL6956071

SCHEMBL6956071

OC(c1ccccc1Cl)c1cc(Cl)ccc1NCC1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FDFT1 P37268 9/20 0.52
CNR1 P21554 6/20 0.44
CNR2 P34972 3/20 0.40
CXCR4 P61073 1/20 0.39
EPHX1 P07099 1/20 0.39
EPHX2 P34913 1/20 0.39
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799234 0.76 FDFT1 (0.42) FDFT1
SCHEMBL7340285 0.76 MAPK1 (0.49) CNR1CNR2EPHX1EPHX2NPC1
SCHEMBL8118267 0.75 FDFT1 (0.48) FDFT1
SCHEMBL6956611 0.75 FDFT1 (0.41) FDFT1
SCHEMBL8799319 0.74 ADRB2 (0.44) FDFT1CNR1
SCHEMBL9727045 0.74 FDFT1 (0.43) FDFT1CNR1
SCHEMBL10886234 0.73 EBP (0.50) CXCR4EPHX1NPC1RAB9A
SCHEMBL8564882 0.69 KDM4E (0.49) FDFT1EPHX1NPC1RAB9A
SCHEMBL8564876 0.69 KDM4E (0.49) FDFT1EPHX1NPC1RAB9A
SCHEMBL11168379 0.69 KDM4E (0.59) CNR1CNR2EPHX1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0567026-B1 4,1-Benzoxazepin derivatives as squalene synthase inhibitors and their use in the treatment of hypercholesteremia and as fungicides TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-26 EP disclosed
EP-0567026-A1 4,1-Benzoxazepin derivatives as squalene synthase inhibitors and their use in the treatment of hypercholesteremia and as fungicides TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-10-27 EP disclosed