SCHEMBL6956404

SCHEMBL6956404

O=C(N[C@@]1([C@H]2CC[C@@H](c3ccccc3O)CC2)CCNC1)N1C(=O)OC[C@@H]1c1ccc(F)c(F)c1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
QPCT Q16769 2/20 0.34
AKT1 P31749 1/20 0.31
ADRA1D P25100 6/20 0.31
ADRA1A P35348 6/20 0.31
ADRA1B P35368 6/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6961569 1.00 QPCT (0.34) QPCTAKT1ADRA1DADRA1AADRA1B
SCHEMBL6965561 0.90 ADRA1A (0.41) QPCTADRA1DADRA1AADRA1B
SCHEMBL6955128 0.90 ADRA1D (0.37) QPCTADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL6967097 0.89 ADRA1D (0.36) QPCTAKT1ADRA1DADRA1AADRA1B
SCHEMBL6958679 0.88 ADRA1A (0.39) QPCTADRA1DADRA1AADRA1B
SCHEMBL6958793 0.87 ADRA1D (0.33) QPCTADRA1DADRA1AADRA1B
SCHEMBL6964803 0.87 ADRA1A (0.40) QPCTADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL6964413 0.86 ADRA1A (0.39) QPCTAKT1ADRA1DADRA1AADRA1B
SCHEMBL6956980 0.85 ADRA1D (0.31) ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL6960279 0.85 ADRA1D (0.31) ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998285-A4 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2003-01-08 EP claimed
EP-0998285-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-05-10 EP claimed
WO-1998057641-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1998-12-23 WO claimed