SCHEMBL6965561

SCHEMBL6965561

N#Cc1ccccc1[C@H]1CC[C@@H]([C@]2(NC(=O)N3C(=O)OC[C@@H]3c3ccc(F)c(F)c3)CCNC2)CC1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 17/20 0.41
ADRA1D P25100 15/20 0.41
ADRA1B P35368 15/20 0.41
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
HRH1 P35367 1/20 0.33
QPCT Q16769 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6956404 0.90 QPCT (0.34) ADRA1AADRA1DADRA1BQPCT
SCHEMBL6961569 0.90 QPCT (0.34) ADRA1AADRA1DADRA1BQPCT
SCHEMBL6955128 0.88 ADRA1D (0.37) ADRA1AADRA1DADRA1BQPCT
Hydrochloric Acid SCHEMBL6967097 0.87 ADRA1D (0.36) ADRA1AADRA1DADRA1BQPCT
SCHEMBL6958679 0.86 ADRA1A (0.39) ADRA1AADRA1DADRA1BADRA2AADRA2B
SCHEMBL6958793 0.85 ADRA1D (0.33) ADRA1AADRA1DADRA1BQPCT
SCHEMBL6964803 0.85 ADRA1A (0.40) ADRA1AADRA1DADRA1BQPCT
Hydrochloric Acid SCHEMBL6964413 0.84 ADRA1A (0.39) ADRA1AADRA1DADRA1BQPCT
SCHEMBL6956980 0.83 ADRA1D (0.31) ADRA1AADRA1DADRA1B
SCHEMBL6955993 0.83 ADRA1A (0.32) ADRA1AADRA1DADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998285-A4 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2003-01-08 EP claimed
EP-0998285-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-05-10 EP claimed
WO-1998057641-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1998-12-23 WO claimed