SCHEMBL6956744

SCHEMBL6956744

N#Cc1ccc(N2CCNCC2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.63
TP53 P04637 1/20 0.63
DRD2 P14416 1/20 0.62
DRD3 P35462 1/20 0.62
ADRB1 P08588 5/20 0.59
HTR3E A5X5Y0 3/20 0.59
HTR3B O95264 3/20 0.59
HTR3A P46098 3/20 0.59
HTR3D Q70Z44 3/20 0.59
HTR3C Q8WXA8 3/20 0.59
SIGMAR1 Q99720 3/20 0.59
ADRB2 P07550 1/20 0.53
NCF1 P14598 1/20 0.53
PLD1 Q13393 1/20 0.53
CHRNA10 Q9GZZ6 1/20 0.53
CHRNA9 Q9UGM1 1/20 0.53
MAPKAPK2 P49137 4/20 0.52
EGLN2 Q96KS0 1/20 0.50
ALDH1A1 P00352 1/20 0.50
LMNA P02545 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL231077 1.00 KDM4E (0.63) KDM4ETP53DRD2DRD3ADRB1
Hydrochloric Acid SCHEMBL23303443 0.98 KDM4E (0.61) KDM4ETP53DRD2DRD3ADRB1
Hydrochloric Acid SCHEMBL376202 0.98 KDM4E (0.61) KDM4ETP53DRD2DRD3ADRB1
SCHEMBL24989037 0.94 KDM4E (0.58) KDM4ETP53DRD2DRD3ADRB1
SCHEMBL4228201 0.93 KDM4E (0.56) KDM4ETP53DRD2DRD3ADRB1
SCHEMBL2384959 0.87 KDM4E (0.80) KDM4ETP53DRD2DRD3CHRNA10
SCHEMBL6718397 0.85 DRD2 (0.53) KDM4ETP53DRD2DRD3ADRB1
Formic Acid Methyl Ester SCHEMBL28330267 0.85 ADRB1 (0.53) KDM4ETP53DRD2DRD3ADRB1
SCHEMBL5570604 0.84 ADRB1 (0.77) KDM4EADRB1HTR3EHTR3BHTR3A
SCHEMBL154178 0.83 KDM4E (0.68) KDM4ETP53CHRNA10CHRNA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1309567-A2 NITROGENOUS HETEROCYCLIC COMPOUNDS Millennium Pharmaceuticals, Inc. (US) 2003-05-14 EP disclosed
WO-2002016360-A2 NITROGENOUS HETEROCYCLIC COMPOUNDS COR THERAPEUTICS, INC. (US) 2002-02-28 WO disclosed