SCHEMBL6956997

SCHEMBL6956997

CC(C)c1nc(CO)n(Cc2cnc3ccccc3c2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FAAH O00519 7/20 0.36
TDP1 Q9NUW8 1/20 0.35
PIK3CD O00329 1/20 0.35
CNR2 P34972 1/20 0.34
ERCC5 P28715 1/20 0.34
FEN1 P39748 1/20 0.34
ITGB2 P05107 4/20 0.34
ICAM1 P05362 4/20 0.34
ITGAL P20701 4/20 0.34
ALOX5AP P20292 1/20 0.33
PDE10A Q9Y233 1/20 0.33
KDR P35968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972940 0.93 FAAH (0.35) FAAHTDP1PIK3CDCNR2ERCC5
SCHEMBL7084086 0.91 TDP1 (0.36) FAAHTDP1PIK3CDCNR2ERCC5
SCHEMBL6968913 0.89 FAAH (0.36) FAAHCNR2ERCC5FEN1ITGB2
SCHEMBL6966848 0.87 TDP1 (0.42) TDP1ALOX5AP
SCHEMBL6966431 0.87 TP53 (0.37) FAAHTDP1PIK3CDCNR2ERCC5
SCHEMBL6969844 0.86 FAAH (0.36) FAAHPIK3CDERCC5FEN1ITGB2
SCHEMBL6960043 0.85 FAAH (0.35) FAAHPIK3CDERCC5FEN1ITGB2
SCHEMBL14002294 0.83 CCR9 (0.32) TDP1
SCHEMBL7083375 0.83 FAAH (0.34) FAAHPIK3CDERCC5FEN1ITGB2
SCHEMBL6972332 0.82 FAAH (0.35) FAAHITGB2ICAM1ITGALALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed