SCHEMBL6957264

SCHEMBL6957264

[CH2]NC(=O)[C@@H](N)Cc1c[nH]cn1

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CSK P41240 1/20 0.32
NLN Q9BYT8 1/20 0.30
CYP3A4 P08684 1/20 0.30
SLC7A5 Q01650 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1070085 0.86 CSK (0.33) CSKNLNCYP3A4SLC7A5
SCHEMBL11620101 0.86 CSK (0.45) CSKNLNCYP3A4SLC7A5
SCHEMBL1070087 0.86 CSK (0.33) CSKNLNCYP3A4SLC7A5
SCHEMBL4197031 0.86 CSK (0.45) CSKNLNCYP3A4SLC7A5
SCHEMBL15292000 0.85 SLC15A1 (0.40) CYP3A4SLC7A5
SCHEMBL3835499 0.84 LTA4H (0.33) CSKNLNCYP3A4SLC7A5
SCHEMBL14151247 0.84 NLN (0.39) NLN
SCHEMBL3835494 0.84 LTA4H (0.33) CSKNLNCYP3A4SLC7A5
SCHEMBL30745117 0.84 CSK (0.32) CSKNLNCYP3A4SLC7A5
SCHEMBL27913327 0.83 CYP3A4 (0.33) CSKNLNCYP3A4SLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757677-B1 BENZOCYCLOHEXYLIMIDAZOLETHIONE DERIVATIVES SYNTEX LLC (US) 2003-06-18 EP disclosed
US-5719280-A REACTING AMINE SUBSTITUTED BENZOCYCLOALKANE WITH DIALKYLOXYACETALDEHYDE IN PRESENCE OF REDUCING AGENT OR CATALYTIC HYDROGENATION, TREATING WITH THIOCYANIC ACID SYNTEX (U.S.A.) INC. (US) 1998-02-17 US disclosed
EP-0757677-A1 BENZOCYCLOALKYLAZOLETHIONE DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1997-02-12 EP disclosed
US-5538988-A CARDIOVASCULAR DISORDERS AND DOPAMINE HYDROLASE ENZYME INHIBITORS SYNTEX (U.S.A.) INC. 1996-07-23 US disclosed
WO-1995029165-A2 BENZOCYCLOALKYLAZ0LETHIONE DERIVATIVES AS DOPAMIN BETA-HYDROXYLASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1995-11-02 WO disclosed